SCHEMBL485838

SCHEMBL485838

CCc1ccc(C2CC(NC(=O)Oc3cncc(Cl)c3)CN(C(=O)C3CCCC3)C2)cc1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
F2R P25116 11/20 0.61
FAAH O00519 3/20 0.36
TACR3 P29371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL661835 0.85 F2R (0.64) F2R
SCHEMBL485888 0.82 F2R (0.65) F2RTACR3
SCHEMBL486466 0.80 F2R (0.69) F2R
SCHEMBL485844 0.79 F2R (0.61) F2R
SCHEMBL486104 0.78 F2R (0.61) F2RFAAH
SCHEMBL662897 0.78 F2R (0.81) F2R
SCHEMBL485980 0.76 F2R (0.73) F2R
SCHEMBL486133 0.76 F2R (1.00) F2R
SCHEMBL662549 0.76 F2R (0.74) F2R
SCHEMBL662802 0.75 F2R (0.67) F2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411363-B1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS BAYER IP GMBH (DE) 2015-10-07 EP disclosed
EP-2411363-A1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS Bayer Pharma AG (DE) 2012-02-01 EP disclosed
WO-2010108608-A1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-09-30 WO disclosed