Pyrazofurin

Pyrazofurin

SCHEMBL4861

NC(=O)c1[nH]nc(C2OC(CO)C(O)C2O)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
UMPS P11172 2/20 1.00
PYGL P06737 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
BLM P54132 1/20 0.39
HIF1A Q16665 1/20 0.38
LMNA P02545 3/20 0.37
GLA P06280 1/20 0.37
EIF4E P06730 1/20 0.37
CYP3A4 P08684 1/20 0.37
TOP1 P11387 1/20 0.37
ADORA1 P30542 1/20 0.37
THPO P40225 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrazofurin SCHEMBL21392925 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11835057 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11826269 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL27539623 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11835064 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL4860 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL29370114 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11726623 0.99 UMPS (0.97) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL10584948 0.95 UMPS (0.90) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
SCHEMBL11826483 0.78 UMPS (0.63) UMPSALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11338 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2026-05-28 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-4705284-A1 4'-HALOGEN CONTAINING NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO Emory University (US) 2026-03-11 EP claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
WO-2025235664-A1 PURINE NUCLEOTIDE AND NUCLEOSIDE THERAPEUTIC COMPOSITIONS AND USES RELATED THERETO EMORY UNIVERSITY (US) 2025-11-13 WO claimed
US-20250268993-A1 ALKALINE PHOSPHATE-BASED ONCOLOGY TREATMENTS THERIVA BIOLOGICS, INC. 2025-08-28 US claimed
US-12318434-B2 Alkaline phosphate-based oncology treatments THERIVA BIOLOGICS, INC. (US) 2025-06-03 US claimed
US-12268694-B2 Combination pharmaceutical agents as RSV inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2025-04-08 US claimed
EP-4524131-A1 SMALL MOLECULES FOR TREATING CANCER, INHABITING CHEMOKINE ACTIVITY AND/OR INDUCING CELL DEATH AlonBio Ltd. (IL) 2025-03-19 EP claimed
US-12202803-B2 Small molecules for treating cancer, inhibiting chemokine activity and/or inducing cell death ALONBIO LTD. (IL) 2025-01-21 US claimed
EP-0594667-A4 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO NEURON INC (US) 1996-01-10 EP claimed
WO-1994026761-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1994-11-24 WO claimed
EP-0594667-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1994-05-04 EP claimed
CN-1071577-A Handle the toxicity of chemotherapy reagent and Anti-virus agent with acylated pyrimidine nucleosides PRO NEURON INC (US) 1993-05-05 CN claimed
WO-1993001202-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1993-01-21 WO claimed
EP-0500586-A4 PYRIMIDINE BIOSYNTHESIS INHIBITORS USEFUL AS IMMUNOSUPPRESSIVE AGENTS 1992-11-04 EP claimed
EP-0500586-A1 PYRIMIDINE BIOSYNTHESIS INHIBITORS USEFUL AS IMMUNOSUPPRESSIVE AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-09-02 EP claimed
US-5102883-A Treating autoimmune diseases, antiinflammatory agent and organ transplantation rejection DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1992-04-07 US claimed
WO-1991006863-A1 PYRIMIDINE BIOSYNTHESIS INHIBITORS USEFUL AS IMMUNOSUPPRESSIVE AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1991-05-16 WO claimed
US-4053698-A ACYLATION OF PYRAZOFURIN ELI LILLY AND COMPANY (US) 1977-10-11 US claimed