Pyrazofurin

Pyrazofurin

SCHEMBL21392925

NC(=O)c1[nH]nc([C@@H]2O[C@H](CO)C(O)C2O)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
UMPS P11172 2/20 1.00
PYGL P06737 5/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
BLM P54132 1/20 0.39
HIF1A Q16665 1/20 0.38
LMNA P02545 3/20 0.37
GLA P06280 1/20 0.37
EIF4E P06730 1/20 0.37
CYP3A4 P08684 1/20 0.37
TOP1 P11387 1/20 0.37
ADORA1 P30542 1/20 0.37
THPO P40225 1/20 0.37
PMP22 Q01453 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrazofurin SCHEMBL11835057 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11826269 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL27539623 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11835064 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL4860 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL4861 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL29370114 1.00 UMPS (1.00) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL11726623 0.99 UMPS (0.97) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
Pyrazofurin SCHEMBL10584948 0.95 UMPS (0.90) UMPSPYGLSMN1; SMN2ALDH1A1TSHR
SCHEMBL11826483 0.78 UMPS (0.63) UMPSALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220218731-A1 COMBINATION THERAPIES FOR CANCER TREATMENT CLEAR CREEK BIO INC (US) 2022-07-14 US disclosed
US-20210315880-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS CLEAR CREEK BIO INC (US) 2021-10-14 US disclosed
US-20210308117-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS CLEAR CREEK BIO INC (US) 2021-10-07 US disclosed
US-20210290651-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS CLEAR CREEK BIO INC (US) 2021-09-23 US disclosed
US-20190290635-A1 METHODS OF TREATING BRAIN CANCER USING AGENTS THAT ALTER ACTIVITY OF A METABOLIC PATHWAY Clear Creek Bio, Inc. 2019-09-26 US disclosed
US-20190290892-A1 METHODS OF DETERMINING DOSING OF A THERAPEUTIC AGENT BASED ON MEASURED LEVELS OF A METABOLITE Clear Creek Bio, Inc. 2019-09-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210315880-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS DHODH, DHFR, DPYD UMPS 64/4885PYGL 2456/4885SMN1; SMN2 2783/4885
US-20190290635-A1 METHODS OF TREATING BRAIN CANCER USING AGENTS THAT ALTER ACTIVITY OF A METABOLIC PATHWAY DHODH, IDH2, DLD UMPS 796/4885PYGL 1747/4885SMN1; SMN2 3467/4885
US-20210290651-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS DHODH, DHFR, DPYD UMPS 64/4885PYGL 2456/4885SMN1; SMN2 2783/4885
US-20210308117-A1 METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS DHODH, DHFR, DPYD UMPS 64/4885PYGL 2456/4885SMN1; SMN2 2783/4885
US-20220218731-A1 COMBINATION THERAPIES FOR CANCER TREATMENT PCK2, PC, FOLR2 UMPS 1839/4885PYGL 871/4885SMN1; SMN2 4169/4885
US-20190290892-A1 METHODS OF DETERMINING DOSING OF A THERAPEUTIC AGENT BASED ON MEASURED LEVELS OF A METABOLITE IDH2, NQO1, TXNRD2 UMPS 1605/4885PYGL 780/4885SMN1; SMN2 1573/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.