SCHEMBL4862357

SCHEMBL4862357

N=C(Nc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
MEN1 O00255 6/20 0.54
KMT2A Q03164 6/20 0.54
POLB P06746 3/20 0.54
TDP1 Q9NUW8 1/20 0.54
NOX1 Q9Y5S8 1/20 0.52
KCNK3 O14649 1/20 0.46
KCNK9 Q9NPC2 1/20 0.46
MITF O75030 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
CYP2C9 P11712 1/20 0.45
EGFR P00533 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
LMNA P02545 2/20 0.44
RECQL P46063 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28624148 0.92 MEN1 (0.54) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL393417 0.85 ALDH1A1 (0.48) NPC1RAB9AMEN1KMT2ANOX1
SCHEMBL457388 0.83 ALDH1A1 (0.46) NPC1RAB9AMEN1KMT2ANOX1
Hydrochloric Acid SCHEMBL9773792 0.83 ALDH1A1 (0.46) NPC1RAB9AMEN1KMT2ANOX1
SCHEMBL19937963 0.82 GAA (0.53) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL14223698 0.81 PTPN1 (0.44) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL14223446 0.81 PTPN1 (0.44) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL4854779 0.81 KMT2A (0.58) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL6960874 0.80 MEN1 (0.55) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL4853047 0.80 NPC1 (0.61) NPC1RAB9AMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264899-B 1,3,5-oxadiazine compound and preparation and application thereof 台州学院 2022-06-14 CN disclosed
CN-113264899-A 1,3,5-oxadiazine compound and preparation and application thereof 台州学院 2021-08-17 CN disclosed
CN-111533706-B Preparation method of 1,4, 6-trisubstituted 1, 2-dihydro-triazine compound 台州学院 2021-08-03 CN disclosed
CN-111533706-A Preparation method of 1,4, 6-trisubstituted 1, 2-dihydro-triazine compound 台州学院 2020-08-14 CN disclosed
CN-106946790-B A kind of preparation method of 1,2- substituted benzimidazole analog derivative 华侨大学 2019-08-06 CN disclosed
CN-108084110-A 3- amino benzo [d] isothiazole, derivative and its synthetic method 湘潭大学 2018-05-29 CN disclosed
CN-106946790-A A kind of preparation method of 1,2 substituted benzimidazole analog derivative 华侨大学 2017-07-14 CN disclosed
US-7365069-B2 Pyrimidone derivatives BEXEL PHARMACEUTICALS INC. (US) 2008-04-29 US disclosed
US-7365069-B2 Pyrimidone derivatives BEXEL PHARMACEUTICALS INC. (US) 2008-04-29 US disclosed
US-7365069-B2 Pyrimidone derivatives BEXEL PHARMACEUTICALS INC. (US) 2008-04-29 US disclosed
US-20040259891-A1 Novel pyrimidon derivatives ORCHID CHEMICAL & PHARMACEUTICALS LIMITED (IN) 2004-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040259891-A1 Novel pyrimidon derivatives TYMS, TPMT, TYMP NPC1 1563/4885RAB9A 2079/4885MEN1 917/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.