SCHEMBL457388

SCHEMBL457388

N=C(Nc1ccccc1)c1ccccc1.[NaH]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.46
TAS2R38 P59533 3/20 0.46
HSD17B10 Q99714 3/20 0.46
TP53 P04637 2/20 0.46
TSHR P16473 2/20 0.46
EPHX1 P07099 2/20 0.46
EPHX2 P34913 1/20 0.46
CDK9 P50750 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
CYP3A4 P08684 1/20 0.46
MEN1 O00255 3/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
KMT2A Q03164 3/20 0.45
SIRT1 Q96EB6 1/20 0.45
PTPN1 P18031 3/20 0.44
GAA P10253 2/20 0.43
NOX1 Q9Y5S8 1/20 0.43
TYR P14679 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL393417 0.98 ALDH1A1 (0.48) ALDH1A1TAS2R38HSD17B10TP53TSHR
Hydrochloric Acid SCHEMBL9773792 0.95 ALDH1A1 (0.46) ALDH1A1TAS2R38HSD17B10TP53TSHR
SCHEMBL19937963 0.85 GAA (0.53) ALDH1A1TP53MEN1NPC1RAB9A
SCHEMBL12755248 0.85 PTPN1 (0.57) ALDH1A1SMN1; SMN2MEN1NPC1RAB9A
SCHEMBL4853047 0.83 NPC1 (0.61) ALDH1A1SMN1; SMN2MEN1NPC1RAB9A
SCHEMBL5779983 0.83 JAK2 (0.61) ALDH1A1EPHX1SMN1; SMN2CYP3A4MEN1
SCHEMBL28624148 0.83 MEN1 (0.54) ALDH1A1SMN1; SMN2CYP3A4MEN1NPC1
SCHEMBL4862357 0.83 NPC1 (0.61) ALDH1A1SMN1; SMN2MEN1NPC1RAB9A
SCHEMBL2154879 0.83 NPC1 (0.52) ALDH1A1TAS2R38HSD17B10TP53SMN1; SMN2
SCHEMBL13437648 0.83 MAOA (0.55) ALDH1A1TP53EPHX1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9630928-B2 Intermediates to prepare herbicidal pyrimidone derivatives E. I. DU PONT DE NEMOURS AND COMPANY (US) 2017-04-25 US disclosed
EP-2475654-B1 HERBICIDAL PYRIMIDONE DERIVATIVES DU PONT (US) 2016-12-28 EP disclosed
US-20160024020-A1 INTERMEDIATES TO PREPARE HERBICIDAL PYRIMIDONE DERIVATIVES FMC CORPORATION 2016-01-28 US disclosed
US-9187432-B2 Intermediates to prepare herbicidal pyrimidone derivatives E I DU PONT DE NEMOURS AND COMPANY (US) 2015-11-17 US disclosed
US-20150105549-A1 INTERMEDIATES TO PREPARE HERBICIDAL PYRIMIDONE DERIVATIVES FMC CORPORATION 2015-04-16 US disclosed
US-8952024-B2 Herbicidal pyrimidone derivatives E I DU PONT DE NEMOURS AND COMPANY (US) 2015-02-10 US disclosed
EP-2475654-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. du Pont de Nemours and Company (US) 2012-07-18 EP disclosed
US-20120149573-A1 HERBICIDAL BUS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES FMC CORPORATION 2012-06-14 US disclosed
WO-2012033548-A2 HERBICIDAL BIS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-15 WO disclosed
WO-2011031658-A1 HERBICIDAL PYRIMIDONE DERIVATIVES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2011-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120149573-A1 HERBICIDAL BUS-NITROGEN-CONTAINING OXO AND SULFONO HETEROCYCLES CBR3, CYP1B1, CBR1 ALDH1A1 1886/4885TAS2R38 2756/4885HSD17B10 629/4885
US-20150105549-A1 INTERMEDIATES TO PREPARE HERBICIDAL PYRIMIDONE DERIVATIVES CBR3, CBR1, MSRB3 ALDH1A1 1015/4885TAS2R38 2734/4885HSD17B10 1461/4885
US-20160024020-A1 INTERMEDIATES TO PREPARE HERBICIDAL PYRIMIDONE DERIVATIVES CBR3, CBR1, PNPO ALDH1A1 830/4885TAS2R38 3152/4885HSD17B10 1358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.