SCHEMBL4863291

SCHEMBL4863291

C=CCOC(=O)c1sc2ccccc2c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
MAOB P27338 4/20 0.47
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 7/20 0.46
TSHR P16473 3/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPT P10636 8/20 0.44
KMT2A Q03164 7/20 0.44
MEN1 O00255 5/20 0.44
MAPK1 P28482 4/20 0.44
LMNA P02545 4/20 0.43
RAB9A P51151 4/20 0.43
GAA P10253 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 3/20 0.43
ALOX15 P16050 2/20 0.43
MAOA P21397 1/20 0.43
NOD2 Q9HC29 1/20 0.41
GLA P06280 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4633547 0.81 ALDH1A1 (0.63) MAOBKDM4EALDH1A1TSHRHSD17B10
SCHEMBL4863286 0.79 CYP3A4 (0.54) CYP3A4KDM4EALDH1A1TSHRHSD17B10
SCHEMBL9660322 0.78 NMT1 (0.57) MAOBKDM4EALDH1A1TSHRMAPT
SCHEMBL4787535 0.76 CYP3A4 (0.47) CYP3A4KDM4EALDH1A1TSHRHSD17B10
SCHEMBL6688219 0.76 ALDH1A1 (0.51) CYP3A4KDM4EALDH1A1TSHRHSD17B10
SCHEMBL3205728 0.76 KDM4E (0.42) CYP3A4MAOBKDM4EALDH1A1HSD17B10
SCHEMBL4651653 0.75 MAPK1 (0.71) MAOBKDM4EALDH1A1TSHRHSD17B10
SCHEMBL31347574 0.75 MAPK1 (0.71) MAOBKDM4EALDH1A1TSHRHSD17B10
SCHEMBL31232901 0.73 ALDH1A1 (0.41) CYP3A4KDM4EALDH1A1TSHRHSD17B10
SCHEMBL11799224 0.72 CYP3A4 (0.65) CYP3A4KDM4EALDH1A1TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1972624-A1 Benzoxazinones and their use as ultraviolet light absorbers Clariant International Ltd. (CH) 2008-09-24 EP disclosed
US-3976780-A Methods of protection against emesis in mammals by administration of a 3-alkoxy-thianaphthene-2-carboxamide SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES L'ILE-DE-FRANCE (FR) 1976-08-24 US disclosed
US-3954748-A ANTIEMETICS SOCIETE D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES DE L'ILE-DE-FRANCE (FR) 1976-05-04 US disclosed