SCHEMBL4863501

SCHEMBL4863501

CCn1c(-c2cnn(-c3ccccc3)c2)c([N+](=O)[O-])c(=O)n(CC)c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.46
ADORA2A P29274 5/20 0.46
ADORA2B P29275 5/20 0.46
ADORA1 P30542 5/20 0.46
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
HTT P42858 2/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 1/20 0.43
MITF O75030 1/20 0.43
AGTR1 P30556 1/20 0.43
RAB9A P51151 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TLR9 Q9NR96 1/20 0.43
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
HPGD P15428 2/20 0.38
CFTR P13569 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4866073 0.94 ADORA2B (0.55) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4863931 0.88 ADORA2A (0.44) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4868150 0.88 HSP90AA1 (0.43) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4868526 0.87 ADORA2B (0.50) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4866000 0.87 HSP90AA1 (0.47) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4866210 0.84 ADORA2B (0.45) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4859903 0.84 HSP90AA1 (0.44) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4863923 0.83 ADORA2A (0.51) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4866844 0.83 ADORA1 (0.44) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1
SCHEMBL4864054 0.83 HSP90AA1 (0.43) HSP90AA1ADORA2AADORA2BADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449473-B2 Substituted pyrrolo[3,2-d]pyrimidin-2,4-diones as A2b adenosine receptor antagonists CV THERAPEUTICS, INC. (US) 2008-11-11 US disclosed
US-20050119287-A1 A2B adenosine receptor antagonists GILEAD PALO ALTO, INC. 2005-06-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050119287-A1 A2B adenosine receptor antagonists ADORA2B, ADORA2A, ADORA3 HSP90AA1 1863/4885ADORA2A 2/4885ADORA2B 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.