SCHEMBL4864185

SCHEMBL4864185

N#CC[C@]1(C(=O)O)CC[C@@H](c2ccccc2OCc2ccccc2)N1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
ALDH1A1 P00352 1/20 0.39
SGMS2 Q8NHU3 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PTGS2 P35354 1/20 0.38
TNKS2 Q9H2K2 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
FFAR2 O15552 1/20 0.36
PPIA P62937 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
FAAH O00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2839962 0.84 KCNH2 (0.43) ALDH1A1SMN1; SMN2
SCHEMBL2834210 0.84 KCNH2 (0.43) ALDH1A1SMN1; SMN2
SCHEMBL2831509 0.81 KCNH2 (0.46) ALDH1A1POLBTNKS2SIRT1FAAH
SCHEMBL4830206 0.80 HTR1A (0.46) HTR1ASLC6A2SLC6A4SLC6A3MEN1
SCHEMBL2835604 0.74 GUSB (0.43) ALDH1A1SMN1; SMN2
SCHEMBL2834323 0.72 KCNH2 (0.52) FFAR2
SCHEMBL11662303 0.69 HTR1A (0.48) HTR1ASLC6A2SLC6A4SLC6A3MEN1
SCHEMBL2835553 0.67 SCN3A (0.49) FFAR2
SCHEMBL4710269 0.66 FFAR2 (0.51) HTR1ASLC6A2SLC6A4SLC6A3MEN1
SCHEMBL4637674 0.66 FFAR2 (0.51) HTR1ASLC6A2SLC6A4SLC6A3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934176-A1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LIMITED (GB) 2008-06-25 EP disclosed
WO-2007042240-A1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LIMITED (GB) 2007-04-19 WO disclosed