SCHEMBL4865743

SCHEMBL4865743

O=S(=O)(c1cccc(Cl)c1)c1ccc2c(c1)CCC2NC1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 13/20 0.47
HTR2C P28335 5/20 0.47
HTR2B P41595 4/20 0.47
HTR1A P08908 2/20 0.47
HTR1D P28221 2/20 0.47
HTR1B P28222 2/20 0.47
HTR7 P34969 2/20 0.47
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
FADS1 O60427 1/20 0.39
WNT3 P56703 1/20 0.39
SFRP1 Q8N474 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3853169 0.90 HTR2C (0.53) HTR6HTR2CHTR2BWNT3SFRP1
SCHEMBL3857911 0.83 HTR6 (0.55) HTR6HTR2CHTR2BWNT3SFRP1
SCHEMBL3844022 0.76 HTR6 (0.54) HTR6HTR2CHTR2BCYP3A4
SCHEMBL1012930 0.72 HTR6 (0.56) HTR6
SCHEMBL13989700 0.71 HTR2C (0.55) HTR6HTR2CHTR2BHTR1B
SCHEMBL5690967 0.71 PDPK1 (0.54) HTR6HTR2CHTR1BFADS1CA1
Hydrochloric Acid SCHEMBL4901126 0.70 HTR2C (0.54) HTR6HTR2CHTR2BHTR1AHTR1D
SCHEMBL14437278 0.70 CNR1 (0.49) HTR6HTR2BPDE4APDE4BPDE4C
SCHEMBL27752358 0.68 HTR6 (0.58) HTR6
SCHEMBL315805 0.68 HTR6 (0.80) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008524274-A 2008-07-10 JP claimed
EP-1831189-A1 TETRALIN AND INDANE DERIVATIVES AND USES THEREOF F. Hoffmann-Roche AG (CH) 2007-09-12 EP claimed
WO-2006066745-A1 TETRALIN AND INDANE DERIVATIVES AND USES THEREOF F.HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO claimed