SCHEMBL4865816

SCHEMBL4865816

Nc1cccc(CN(C(=O)Nc2ccccc2)N(Cc2cccc([N+](=O)[O-])c2)C(=O)Nc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KMT2A Q03164 6/20 0.49
MEN1 O00255 5/20 0.49
LMNA P02545 2/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
MAPT P10636 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
BAZ1A Q9NRL2 1/20 0.46
DDX3X O00571 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
CTDSP1 Q9GZU7 1/20 0.45
THRB P10828 1/20 0.45
HPGD P15428 1/20 0.45
ALOX12 P18054 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865811 0.81 NAMPT (0.65) ALDH1A1SMN1; SMN2KMT2AMEN1NPC1
Hydrochloric Acid SCHEMBL4856345 0.77 ALDH1A1 (0.53) ALDH1A1SMN1; SMN2KMT2AMEN1LMNA
SCHEMBL4864537 0.77 CYP2D6 (0.46) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL11144060 0.76 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2KMT2AMEN1NPC1
SCHEMBL13623020 0.75 ALDH1A1 (0.74) ALDH1A1SMN1; SMN2KMT2AMEN1LMNA
SCHEMBL10160140 0.74 ALDH1A1 (0.86) ALDH1A1SMN1; SMN2KMT2AMEN1LMNA
Hydrochloric Acid SCHEMBL1026974 0.74 ALDH1A1 (0.72) ALDH1A1SMN1; SMN2KMT2AMEN1LMNA
Trifluoroacetic Acid SCHEMBL1026824 0.73 ALDH1A1 (0.67) ALDH1A1SMN1; SMN2KMT2AMEN1LMNA
Trifluoroacetic Acid SCHEMBL1074988 0.73 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2KMT2AMEN1MAPT
SCHEMBL4866357 0.72 MEN1 (0.67) ALDH1A1SMN1; SMN2KMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7384963-B2 2′-Methyl-5-(1,3,4-oxadiazol-2-yl)1, 1′-biphenyl-4-carboxaide derivatives and their use as p38 kinase GLAXO GROUP LIMITED (GB) 2008-06-10 US disclosed