SCHEMBL4868057

SCHEMBL4868057

COc1ccc(CC2(N)CCCC2)cc1.Nc1ccc(C(N)C2CCCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 4/20 0.40
SLC6A3 Q01959 3/20 0.40
SLC6A2 P23975 2/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDE4A P27815 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP3A4 P08684 1/20 0.36
EPHX2 P34913 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4868046 0.84 TDP1 (0.52) SLC6A4SLC6A3TDP1MAPK1ALDH1A1
SCHEMBL1822033 0.78 MAOB (0.47) SLC6A4SLC6A3
SCHEMBL14390178 0.78 SLC6A4 (0.54) SLC6A4SLC6A3SLC6A2CYP1A2CYP2D6
SCHEMBL1824988 0.77 SLC6A4 (0.46) SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL3966019 0.77 IDO1 (0.47) SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL3967323 0.76 IDO1 (0.46) SLC6A4SLC6A3SLC6A2
SCHEMBL297343 0.72 OPRM1 (0.51) SLC6A4SLC6A3SLC6A2CYP1A2CYP2D6
SCHEMBL1824702 0.72 MAOB (0.55) SLC6A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL3964601 0.72 IDO1 (0.36) SLC6A4SLC6A3SLC6A2ALDH1A1RAB9A
SCHEMBL1820867 0.72 MAOB (0.54) TDP1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423035-B2 Substituted cycloalkyl derivatives, process for the manufacture thereof and use thereof as medicament BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-09-09 US disclosed
US-20050261286-A1 Substituted cycloalkyl derivatives, process for the manufacture thereof and use thereof as medicament BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050261286-A1 Substituted cycloalkyl derivatives, process for the manufacture thereof and use thereof as medicament CHRM1, CHRM2, CHRM3 SLC6A4 4448/4885SLC6A3 4799/4885SLC6A2 4781/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.