SCHEMBL4868075

SCHEMBL4868075

CSCCOC(=O)Nc1ncnc2c1ncn2N(CCNS(=O)(=O)c1nc2ccccc2s1)CC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
NFKB1 P19838 1/20 0.33
CYP2C19 P33261 1/20 0.33
STAT1 P42224 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
CA1 P00915 6/20 0.31
CA2 P00918 6/20 0.31
CA4 P22748 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4838306 0.87 PDE4A (0.32) NPC1RAB9ASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL4868081 0.83 CA1 (0.33) ALDH1A1CA1CA2CA4
SCHEMBL3253725 0.82 SMN1; SMN2 (0.33) NPC1RAB9ASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL4835790 0.75 MEN1 (0.34)
SCHEMBL4838731 0.74 PKM (0.34) NPC1RAB9ASMN1; SMN2ALDH1A1NFKB1
SCHEMBL4838681 0.73 ABL1 (0.34) NPC1RAB9AALDH1A1
SCHEMBL4838426 0.73 PDE4A (0.32)
SCHEMBL4842968 0.72 MAPT (0.37) NPC1RAB9ASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL4838348 0.71 GALR3 (0.36) NPC1RAB9ASMN1; SMN2ALDH1A1CYP1A2
SCHEMBL3136422 0.71 MAPK1 (0.32) NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7411065-B2 Peptide nucleic acid monomers: diphenylmethyl, benzyl, alkylthioalkyl, or phenylthioalkyl esters of N-(1-[4-(2-benzothiazolyl-, 2-benzoxazolyl-, 2-benzofuranyl- or 2-benzothiophenyl-sulfonyl)-3-piperazinon-1-ylcarbonylmethyl]pyrimidon-4-yl)carbamic acids PANAGENE, INC. (KR) 2008-08-12 US disclosed