SCHEMBL4868081

SCHEMBL4868081

CSCCOC(=O)c1nc(N)c2ncn(N(CCNS(=O)(=O)c3nc4ccccc4s3)CC(=O)O)c2n1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.33
CA2 P00918 10/20 0.33
CA4 P22748 2/20 0.32
ALDH1A1 P00352 1/20 0.30
CHKA P35790 1/20 0.30
CHKB Q9Y259 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4868075 0.83 NPC1 (0.33) CA1CA2CA4ALDH1A1
SCHEMBL4838306 0.72 PDE4A (0.32) CA1CA2CA4ALDH1A1
SCHEMBL4835790 0.71 MEN1 (0.34)
SCHEMBL4865415 0.69 PKM (0.37) CA1CA2ALDH1A1
SCHEMBL4842968 0.68 MAPT (0.37) CA1CA2CA4ALDH1A1
SCHEMBL3253725 0.67 SMN1; SMN2 (0.33) ALDH1A1
SCHEMBL3138127 0.66 MEN1 (0.34) ALDH1A1
SCHEMBL3140234 0.65 PAX8 (0.42) CA1CA2CA4ALDH1A1
SCHEMBL4865411 0.64 ABL1 (0.41) ALDH1A1
SCHEMBL3137660 0.63 MAPT (0.37) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7411065-B2 Peptide nucleic acid monomers: diphenylmethyl, benzyl, alkylthioalkyl, or phenylthioalkyl esters of N-(1-[4-(2-benzothiazolyl-, 2-benzoxazolyl-, 2-benzofuranyl- or 2-benzothiophenyl-sulfonyl)-3-piperazinon-1-ylcarbonylmethyl]pyrimidon-4-yl)carbamic acids PANAGENE, INC. (KR) 2008-08-12 US disclosed