SCHEMBL4869626

SCHEMBL4869626

COc1ccc2c(c1)CCCCN2C(=O)Nc1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.69
ALDH1A1 P00352 2/20 0.68
L3MBTL1 Q9Y468 2/20 0.68
MAPK1 P28482 1/20 0.68
SMN1; SMN2 Q16637 3/20 0.61
NPC1 O15118 2/20 0.61
PKM P14618 2/20 0.61
NFKB1 P19838 2/20 0.61
RAB9A P51151 2/20 0.61
NFKB2 Q00653 2/20 0.61
RELA Q04206 2/20 0.61
MAOB P27338 1/20 0.61
LMNA P02545 4/20 0.61
TP53 P04637 2/20 0.61
HSD17B10 Q99714 1/20 0.60
THRB P10828 1/20 0.59
NOTUM Q6P988 1/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4863193 0.89 MAPT (0.64) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4869965 0.89 MAPT (0.64) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4860848 0.89 MAPT (0.61) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4869061 0.88 MAPT (0.63) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4870033 0.85 MAPT (0.93) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4870805 0.85 HTR2A (0.63) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4865371 0.85 MAPT (0.58) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL4870653 0.84 PDK1 (0.61) MAPTSMN1; SMN2NPC1PKMNFKB1
SCHEMBL4866075 0.84 TP53 (0.59) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2
SCHEMBL2776090 0.83 HSD17B10 (0.71) MAPTALDH1A1L3MBTL1MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050101600-A1 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 US claimed
EP-1475368-A1 N-CARBAMOYL NITROGEN-CONTAINING FUSED RING COMPOUNDS AND DRUGS CONTAINING THESE COMPOUNDS AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2004-11-10 EP claimed
US-7368444-B2 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-05-06 US disclosed
US-7368444-B2 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-05-06 US disclosed
US-7368444-B2 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-05-06 US disclosed
US-20050101600-A1 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 US disclosed
EP-1475368-A1 N-CARBAMOYL NITROGEN-CONTAINING FUSED RING COMPOUNDS AND DRUGS CONTAINING THESE COMPOUNDS AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2004-11-10 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050101600-A1 N-carbamoyl nitrogen-containing fused ring compounds and drugs containing these compounds as the active ingredient CNR1, CNR2, NPSR1 MAPT 3398/4885ALDH1A1 3990/4885L3MBTL1 4626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.