SCHEMBL4873741

SCHEMBL4873741

COc1cc(CBr)ccc1Cl.Cc1ccc(Cl)c(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
HPGD P15428 3/20 0.46
L3MBTL1 Q9Y468 3/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
MAPK1 P28482 2/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 2/20 0.46
USP2 O75604 1/20 0.46
POLB P06746 1/20 0.46
ALOX12 P18054 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
HSP90AA1 P07900 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GAA P10253 1/20 0.40
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3867553 0.85 MAPT (0.56) MAPTHPGDL3MBTL1CYP2C9CYP2C19
SCHEMBL30029152 0.84 ALDH1A1 (0.47) MAPTHPGDL3MBTL1CYP2C9CYP2C19
SCHEMBL364121 0.84 ALDH1A1 (0.47) MAPTHPGDL3MBTL1CYP2C9CYP2C19
SCHEMBL11651990 0.76 TSHR (0.50) HPGDALDH1A1CYP4F2CYP4A11CYP3A4
SCHEMBL5443737 0.74 TAAR1 (0.65) MAPK1ALDH1A1ALOX12GAACYP3A4
SCHEMBL128701 0.74 MAPT (0.67) MAPTHPGDL3MBTL1CYP2C9CYP2C19
SCHEMBL12002 0.74
SCHEMBL27570328 0.72 TRPA1 (0.56) MAPTHPGDMEN1ALDH1A1KMT2A
SCHEMBL1548047 0.71 NPC1 (0.53) MAPTHPGDL3MBTL1CYP2C9CYP2C19
SCHEMBL6401380 0.71 CYP1A2 (0.62) MEN1KMT2AALOX12GAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937632-A1 NOVEL COMPOUNDS Astra Zeneca AB (SE) 2008-07-02 EP disclosed
WO-2007039736-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2007-04-12 WO disclosed