SCHEMBL4875336

SCHEMBL4875336

O=C(N1CCCCC12CCNCC2)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.35
CNR2 P34972 1/20 0.34
CYP1A2 P05177 1/20 0.33
CA2 P00918 1/20 0.32
CHKA P35790 1/20 0.32
MGLL Q99685 2/20 0.31
ADRA2C P18825 1/20 0.31
JAK1 P23458 1/20 0.30
SOS1 Q07889 1/20 0.30
SOS2 Q07890 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18320297 0.79 NAMPT (0.38) NAMPTCNR2CYP1A2CA2CHKA
SCHEMBL9978112 0.78
Hydrochloric Acid SCHEMBL20135742 0.77 NAMPT (0.37) NAMPTCNR2CYP1A2CA2CHKA
Trifluoroacetic Acid SCHEMBL31579460 0.75 NAMPT (0.34) NAMPTJAK1SOS1SOS2
SCHEMBL15286428 0.73 JAK3 (0.46) NAMPT
SCHEMBL700399 0.73 NAMPT (0.41) NAMPTCNR2CYP1A2CA2CHKA
SCHEMBL799357 0.72 SOS1 (0.35) SOS1SOS2
Hydrochloric Acid SCHEMBL15288269 0.72 JAK3 (0.45) NAMPT
SCHEMBL30875892 0.72 NAMPT (0.40) NAMPTCNR2CYP1A2CA2CHKA
SCHEMBL22208191 0.72 EPHX1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8735411-B2 Macrocyclic benzofused pyrimidine derivatives ABBVIE INC. (US) 2014-05-27 US disclosed
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives ABBVIE INC. 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives DPYD, TYMS, UMPS NAMPT 20/4885CNR2 3540/4885CYP1A2 930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.