SCHEMBL4877494

SCHEMBL4877494

Nc1nc(Cl)c2c(n1)-c1ccccc1S(=O)(=O)CC2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.39
ADORA2A P29274 5/20 0.38
ADORA1 P30542 4/20 0.38
HRH4 Q9H3N8 3/20 0.37
HRH3 Q9Y5N1 2/20 0.37
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
BCHE P06276 2/20 0.35
EGFR P00533 1/20 0.34
KDR P35968 1/20 0.34
EPHA4 P54764 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
ACHE P22303 1/20 0.33
P2RX7 Q99572 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3R2 O00459 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4875280 0.76 HPGD (0.39) MAPK14ADORA2AADORA1HRH4HRH3
SCHEMBL4877642 0.75 BCHE (0.57) ADORA2AADORA1HRH4HRH3HRH2
SCHEMBL606352 0.75 HRH4 (0.64) HRH4HRH3HRH2HRH1
SCHEMBL3341967 0.72 BCHE (0.59) ADORA2AADORA1HRH4HRH3HRH2
SCHEMBL4872907 0.72 HRH4 (0.48) ADORA2AADORA1HRH4HRH3HRH2
SCHEMBL4874208 0.70 NPY5R (0.43) MAPK14ADORA2AADORA1HRH4HRH3
SCHEMBL4876988 0.69 ADORA2A (0.37) MAPK14ADORA2AADORA1HRH4HRH3
SCHEMBL2675124 0.65 KMT2A (0.46) BCHEKDM4EALDH1A1
SCHEMBL10196638 0.63 KMT2A (0.46) BCHEKDM4E
SCHEMBL15662918 0.63 MAPK14 (0.48) MAPK14ADORA2AADORA1HRH4BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8735411-B2 Macrocyclic benzofused pyrimidine derivatives ABBVIE INC. (US) 2014-05-27 US disclosed
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives ABBVIE INC. 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives DPYD, TYMS, UMPS MAPK14 2653/4885ADORA2A 1517/4885ADORA1 2541/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.