SCHEMBL4877899

SCHEMBL4877899

CC(C)(C)OC(=O)N1CC2(CCCN(Cc3ccccc3)C2)C1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 15/20 0.65
ALDH1A1 P00352 4/20 0.65
CYP3A4 P08684 14/20 0.61
TSHR P16473 8/20 0.61
CYP1A2 P05177 3/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
HPGD P15428 1/20 0.54
USP2 O75604 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31230958 0.93 CYP2D6 (0.62) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL21262272 0.93 CYP2D6 (0.60) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL8044838 0.92 CYP2D6 (0.77) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL8060453 0.91 CYP2D6 (0.72) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL14027002 0.89 CYP2D6 (0.65) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL31230964 0.88 CYP2D6 (0.58) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL19173661 0.88 RORC (0.53) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL17608988 0.87 CYP2D6 (0.64) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL1426231 0.87 CYP2D6 (0.64) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2
SCHEMBL2381460 0.87 CYP2D6 (0.59) CYP2D6ALDH1A1CYP3A4TSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8735411-B2 Macrocyclic benzofused pyrimidine derivatives ABBVIE INC. (US) 2014-05-27 US disclosed
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives ABBVIE INC. 2008-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188452-A1 Macrocyclic Benzofused Pyrimidine Derivatives DPYD, TYMS, UMPS CYP2D6 558/4885ALDH1A1 411/4885CYP3A4 653/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.