SCHEMBL4881789

SCHEMBL4881789

Cc1c(Cl)ccc(N=C=O)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.50
TDP1 Q9NUW8 2/20 0.42
MAPK1 P28482 1/20 0.42
TRPA1 O75762 1/20 0.40
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
CES1 P23141 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11475560 0.84 CYP3A4 (0.55) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL10316759 0.82 CYP3A4 (0.48) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL1969003 0.81 TDP1 (0.47) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL11849090 0.80 CYP3A4 (0.46) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL9063336 0.78 CYP3A4 (0.53) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL17196712 0.78 CYP3A4 (0.44) CYP3A4TDP1TRPA1ALDH1A1HPGD
SCHEMBL9551404 0.78 CYP3A4 (0.50) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL1493105 0.78 TDP1 (0.44) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL29796026 0.78 CYP3A4 (0.50) CYP3A4TDP1MAPK1TRPA1ALDH1A1
SCHEMBL28565927 0.77 CYP3A4 (0.52) CYP3A4TDP1MAPK1TRPA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8754107-B2 Aminopyrrolidines as chemokine receptor antagonists ABBVIE INC. (US) 2014-06-17 US disclosed
US-20080176883-A1 Antiinflammtory, antiproliferative, anticancer agents; (3-Hydroxy-pyrrolidin-1-yl)-(3-trifluoromethyl-7,8-dihydro-5H-[1,6]naphthyridin-6-yl)-methanone ABBVIE INC. 2008-07-24 US disclosed
US-5270302-A Derivatives of tetrapeptides as CCK agonists ABBOTT LABORATORIES (US) 1993-12-14 US disclosed
WO-1991019733-A1 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS ABBOTT LABORATORIES (US) 1991-12-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176883-A1 Antiinflammtory, antiproliferative, anticancer agents; (3-Hydroxy-pyrrolidin-1-yl)-(3-trifluoromethyl-7,8-dihydro-5H-[1,6]naphthyridin-6-yl)-methanone MIF, CCL5, CCR2 CYP3A4 916/4885TDP1 2982/4885MAPK1 237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.