SCHEMBL4883657

SCHEMBL4883657

O=C1c2ccccc2C(=O)N1CCc1cc([AsH2])cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.48
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 1/20 0.40
GLS O94925 1/20 0.40
CHRM5 P08912 1/20 0.39
PARK7 Q99497 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL546449 0.84 CASP3 (0.48) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL7956763 0.82 CASP3 (0.55) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL7957008 0.80 ADRA1D (0.62) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL12475302 0.78 KMT2A (0.46) CASP3CA1CA4ALDH1A1SMN1; SMN2
SCHEMBL15078643 0.73 RXFP1 (0.44) CASP3KDM4EALDH1A1MAPTMEN1
SCHEMBL18669177 0.70 CASP3 (0.52) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL29724090 0.70 CASP3 (0.86) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL1142116 0.70 CASP3 (0.86) CASP3ADRA1DADRA1AADRA1BCA1
SCHEMBL18669003 0.70 CA9 (0.61) CASP3CA1CA2CA9KDM4E
Bromide SCHEMBL22366540 0.69 ADRA1D (0.44) CASP3ADRA1DADRA1AADRA1BGLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957460-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2008-08-20 EP disclosed
WO-2007067444-A1 BICYCLIC COMPOUNDS WITH KINASE INHIBITORY ACTIVITY MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-06-14 WO disclosed