SCHEMBL4884773

SCHEMBL4884773

CCCCC[C@@]1(n2cnc3c(N)ncnc32)O[C@H](CO)[C@@H](O)[C@H]1S

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EHMT1 Q9H9B1 1/20 0.47
ADORA3 P0DMS8 4/20 0.47
ADORA2A P29274 4/20 0.47
GMPS P49915 1/20 0.47
EGFR P00533 1/20 0.47
ERBB2 P04626 1/20 0.47
PI4KA P42356 2/20 0.44
PI4K2B Q8TCG2 2/20 0.44
PI4K2A Q9BTU6 2/20 0.44
PI4KB Q9UBF8 2/20 0.44
SLC28A1 O00337 2/20 0.44
DPP4 P27487 1/20 0.44
MEN1 O00255 1/20 0.44
MAP3K7 O43318 1/20 0.44
SLC28A2 O43868 1/20 0.44
GAPDH P04406 1/20 0.44
MAPK1 P28482 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
STAT6 P42226 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3046312 0.97 ADORA3 (0.48) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL9231750 0.91 ADORA3 (0.49) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL10865960 0.90 ADORA3 (0.48) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL1920532 0.90 ADORA3 (0.48) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL3455187 0.89 ADORA3 (0.51) ADORA3ADORA2AGMPSEGFRERBB2
SCHEMBL29509039 0.88 ADORA3 (0.50) EHMT1ADORA3ADORA2AGMPSEGFR
Phosphoric Acid SCHEMBL15210131 0.87 EHMT1 (0.46) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL5562015 0.85 ADORA2A (0.46) EHMT1ADORA3ADORA2AGMPSEGFR
SCHEMBL29444891 0.85 ADORA3 (0.47) ADORA3ADORA2AGMPSEGFRERBB2
SCHEMBL28229420 0.85 ADORA3 (0.47) ADORA3ADORA2AGMPSEGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348315-B2 Methods of treating heart failure with modified ATP, ADP and AMP compounds THE UNIVERSITY OF CONNECTICUT (US) 2008-03-25 US disclosed
US-20030186929-A1 Methods of treating heart failure with modified ATP, ADP and AMP compounds NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2003-10-02 US disclosed
US-6255292-B1 INCREASING CELLULAR CONTRACTIONS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2001-07-03 US disclosed
US-5712258-A Inotropic ADP and ATP analogues and their pharmaceutical compositions THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-01-27 US disclosed
WO-1996029345-A1 NOVEL INOTROPIC AGENTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1996-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186929-A1 Methods of treating heart failure with modified ATP, ADP and AMP compounds ATP5MF, ATP5MG, ATP2A1 EHMT1 1868/4885ADORA3 31/4885ADORA2A 15/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.