SCHEMBL489020

SCHEMBL489020

CC(Oc1cncc(-c2ccc(N)nc2)c1)c1c(F)ccc(F)c1Cl

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
INPPL1 O15357 12/20 0.88
JAK2 O60674 2/20 0.52
MET P08581 6/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30453362 0.83 MET (0.68) INPPL1JAK2MET
SCHEMBL488367 0.83 MET (0.68) INPPL1JAK2MET
SCHEMBL27650172 0.83 INPPL1 (0.62) INPPL1JAK2MET
SCHEMBL16555527 0.82 INPPL1 (0.60) INPPL1MET
SCHEMBL30453499 0.77 MET (0.78) INPPL1JAK2MET
SCHEMBL488221 0.77 MET (0.78) INPPL1JAK2MET
SCHEMBL13276065 0.75 INPPL1 (0.70) INPPL1JAK2MET
SCHEMBL21044530 0.75 INPPL1 (0.57) INPPL1
SCHEMBL30453624 0.74 JAK2 (0.69) INPPL1JAK2MET
SCHEMBL488375 0.74 JAK2 (0.69) INPPL1JAK2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8106197-B2 Aminoheteroaryl compounds as protein kinase inhibitors PFIZER INC. (US) 2012-01-31 US disclosed
US-20070072874-A1 Aminoheteroaryl compounds as protein kinase inhibitors SUGEN, INC. 2007-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070072874-A1 Aminoheteroaryl compounds as protein kinase inhibitors MET, MAP4K1, MAP4K2 INPPL1 1551/4885JAK2 287/4885MET 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.