Triprolidine

Triprolidine

SCHEMBL4905

Cc1ccc(/C(=C\CN2CCCC2)c2ccccn2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Triprolidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 2/20 1.00
KMT2A Q03164 3/20 1.00
LMNA P02545 2/20 1.00
SLC6A4 P31645 2/20 1.00
ADRA1A P35348 2/20 1.00
OPRK1 P41145 2/20 1.00
MEN1 O00255 2/20 1.00
ADRA2B P18089 2/20 1.00
CHRM1 P11229 1/20 1.00
KCNH2 Q12809 1/20 1.00
ALDH1A1 P00352 1/20 1.00
CYP2D6 P10635 1/20 1.00
TSHR P16473 1/20 1.00
NFKB1 P19838 1/20 1.00
THPO P40225 1/20 1.00
NPSR1 Q6W5P4 2/20 0.97
GMNN O75496 1/20 0.97
BLM P54132 1/20 0.97
PMP22 Q01453 1/20 0.97
PTGS2 P35354 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triprolidine SCHEMBL29631820 1.00 KMT2A (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL4906 1.00 KMT2A (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL3881294 1.00 KMT2A (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL9723510 0.99 LMNA (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL42146 0.99 LMNA (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL3273486 0.99 KMT2A (0.97) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL42145 0.99 LMNA (1.00) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL1140974 0.97 LMNA (0.98) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL1140976 0.97 LMNA (0.98) KMT2ALMNASLC6A4ADRA1AHRH1
Triprolidine SCHEMBL14973526 0.97 KMT2A (0.95) KMT2ALMNASLC6A4ADRA1AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 14979 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4704971-A1 GAMMA STIMULATION AND NEUROMODULATOR COMBINATION THERAPY Cognito Therapeutics, Inc. (US) 2026-03-11 EP claimed
US-12569451-B2 Bio-inspired tissue-adhesive hydrogel patch and uses thereof Cellartgen Inc. (KR) 2026-03-10 US claimed
EP-4691492-A2 LIQUID COMPOSITIONS Kenvue Brands LLC (US) 2026-02-11 EP claimed
EP-4630401-A2 CARBONIC ANHYDRASE ENZYME INHIBITORS AND METHODS OF USE THEREOF Rutgers, the State University of New Jersey (US) 2025-10-15 EP claimed
EP-4247331-B1 ORODISPERSIBLE POWDER COMPOSITION COMPRISING AN ANTIHISTAMINE COMPOUND BIOPHARMA SYNERGIES S L (ES) 2025-10-08 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-20250177398-A1 CARBONIC ANHYDRASE ENZYMES FOR REGULATING MAST CELL HEMATOPOIESIS AND TYPE 2 INFLAMMATION RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2025-06-05 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-12296043-B2 Liquisoft capsules PATHEON SOFTGELS INC. (US) 2025-05-13 US claimed
EP-0063649-B1 NON-INVASIVE MEASURING DEVICE FOR LOCATING DRAINAGE AND CIRCULATION MALFUNCTIONS IN VEINS AND ARTERIES Blazek, Vladimir, Dr.-Ing. (DE) 1985-09-04 EP claimed
EP-0151987-A2 Means for the treatment of diseases of the veins and the anal region Ismail, Roshdy, Dr. (DE) 1985-08-21 EP claimed
WO-1985000982-A1 SYRINGE CONNECTABLE TO A VEIN CATHETER TO CONTROL ITS POSITION DURING ITS SETTING AND UTILIZATION MAERZ PETER 1985-03-14 WO claimed
EP-0117519-A1 Catheter Theermann, Johannes, Dipl.-Ing. (DE) 1984-09-05 EP claimed
EP-0106304-A2 Orthopaedic device Best, Peter (DE) 1984-04-25 EP claimed
EP-0082504-A1 Catheter for the catheterisation of central veins Sterimed Gesellschaft für medizinischen Bedarf mbH (DE) 1983-06-29 EP claimed
WO-1983002064-A1 CATHETER FOR CENTRAL VEINS KRAMANN, BERNHARD 1983-06-23 WO claimed
WO-1983001894-A1 DEVICE FOR ELIMINATING OR EXPANDING STRICTURES IN VESSELS CONDUCTING BODY LIQUIDS WEIKL, ANDREAS 1983-06-09 WO claimed
EP-0063649-A1 Non-invasive measuring device for locating drainage and circulation malfunctions in veins and arteries Blazek, Vladimir, Dr.-Ing. (DE) 1982-11-03 EP claimed
EP-0041696-A1 Blood pressure measuring device Rieckmann, Jutta, Geb. Federlein (DE) 1981-12-16 EP claimed