SCHEMBL490532

SCHEMBL490532

CCCCC(CC)COC(=O)CCc1cc(O)c(O)c(O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.61
TSHR P16473 3/20 0.61
TDP1 Q9NUW8 2/20 0.61
ATM Q13315 1/20 0.61
LMNA P02545 3/20 0.50
ALDH1A1 P00352 5/20 0.48
CA2 P00918 1/20 0.48
MAPK1 P28482 3/20 0.46
RECQL P46063 1/20 0.46
HSD17B10 Q99714 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
BCL2L1 Q07817 1/20 0.40
ESR1 P03372 2/20 0.40
APP P05067 1/20 0.39
CNR2 P34972 1/20 0.38
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223518 0.89 CYP3A4 (0.59) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490663 0.88 CYP3A4 (0.62) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490525 0.88 CYP3A4 (0.58) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490494 0.86 CYP3A4 (0.57) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL284444 0.85 CYP3A4 (0.56) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490725 0.85 CYP3A4 (0.61) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL27205429 0.84 CYP3A4 (0.54) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490573 0.83 CYP3A4 (0.57) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL490538 0.83 CYP3A4 (0.62) CYP3A4TSHRTDP1ATMLMNA
SCHEMBL28675853 0.82 PRSS1 (0.52) CYP3A4TSHRTDP1ATMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8268293-B2 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2012-09-18 US disclosed
US-8106233-B2 Applying di-2-ethylhexyl 4-hydroxy-3,5-dimethoxy-benzylmalonate; protective action against UV rays, oxidative stress on body cells, counters skin ageing MERCK PATENT GMBH (DE) 2012-01-31 US disclosed
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2008-07-17 US disclosed
US-20080152603-A1 Antioxidants SUSONITY Commercial GmbH (DE) 2008-06-26 US disclosed
CN-101203278-A Ultraviolet protection MERCK PATENT GMBH (DE) 2008-06-18 CN disclosed
EP-1871735-A1 ANTIOXIDANTS Merck Patent GmbH (DE) 2008-01-02 EP disclosed
WO-2006111233-A1 ANTIOXIDANTS MERCK PATENT GMBH (DE) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080152603-A1 Antioxidants GPX4, GPX1, CAT CYP3A4 392/4885TSHR 4679/4885TDP1 1049/4885
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives HPD, HAAO, UGT1A6 CYP3A4 63/4885TSHR 4810/4885TDP1 2793/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.