SCHEMBL4906559

SCHEMBL4906559

COC(=O)c1cc(S(=O)(=O)NCCc2nc(-c3ccc4ccccc4c3)sc2C)cc(C)c1C

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 8/20 0.40
MAPT P10636 6/20 0.40
POLB P06746 2/20 0.40
ALDH1A1 P00352 3/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TP53 P04637 6/20 0.39
PLAU P00749 1/20 0.38
KMT2A Q03164 2/20 0.37
HTT P42858 1/20 0.37
MMP3 P08254 1/20 0.36
THRB P10828 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4903767 0.91 LMNA (0.40) LMNAMAPTALDH1A1TP53THRB
SCHEMBL4906115 0.91 POLB (0.46) LMNAMAPTPOLBALDH1A1SLC6A2
SCHEMBL4898005 0.91 MAPT (0.47) LMNAMAPTALDH1A1TP53KMT2A
SCHEMBL4899685 0.89 MAPT (0.42) LMNAMAPTPOLBALDH1A1TP53
SCHEMBL4895407 0.88 MAPT (0.47) LMNAMAPTPOLBALDH1A1TP53
SCHEMBL4901284 0.88 TP53 (0.44) LMNAMAPTALDH1A1TP53KMT2A
SCHEMBL4907641 0.87 PPARA (0.46) LMNAMAPTALDH1A1TP53KMT2A
SCHEMBL4895165 0.86 LMNA (0.40) LMNAMAPTALDH1A1TP53KMT2A
SCHEMBL4906423 0.86 MAPT (0.40) LMNAMAPTTP53
SCHEMBL4900535 0.85 MAPT (0.41) LMNAMAPTPOLBALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PFIZER INC. 2008-04-17 US disclosed
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds HAMANAKA ERNEST S 2006-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060229363-A1 Substituted Heteroaryl- and Phenylsulfamoyl Compounds PPARA, PPARG, PPARD LMNA 317/4885MAPT 1858/4885POLB 1488/4885
US-20080090829-A1 SUBSTITUTED HETEROARYL- AND PHENYLSULFAMOYL COMPOUNDS PPARA, PPARG, PPARD LMNA 319/4885MAPT 1786/4885POLB 1807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.