SCHEMBL4907324

SCHEMBL4907324

N#Cc1cccc(Oc2ncc(Cl)cc2NS(=O)(=O)c2ccc(Cl)s2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 12/20 0.49
PTGER4 P35408 1/20 0.45
PTGER2 P43116 1/20 0.45
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
NFKBIA P25963 2/20 0.43
RELA Q04206 2/20 0.43
PIK3CA P42336 2/20 0.40
MTOR P42345 1/20 0.40
CKS1B P61024 1/20 0.40
SKP2 Q13309 1/20 0.40
MEN1 O00255 1/20 0.40
THRB P10828 1/20 0.40
BLM P54132 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CCR4 P51679 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4913288 0.85 CCR2 (0.69) CCR2PTGER4CYP3A4CYP2C9CYP2C19
SCHEMBL4907421 0.83 CCR2 (0.57) CCR2CYP3A4CYP2C9CYP2C19PIK3CA
SCHEMBL4907638 0.83 CCR2 (0.66) CCR2CYP3A4CYP2C9CYP2C19NFKBIA
SCHEMBL4912558 0.82 CCR2 (0.73) CCR2CYP3A4CYP2C9CYP2C19CCR4
SCHEMBL4912371 0.79 CCR2 (0.54) CCR2CYP3A4CYP2C9CYP2C19CKS1B
SCHEMBL4935740 0.77 CCR2 (0.67) CCR2PTGER4PTGER2CYP3A4CYP2C9
SCHEMBL14006392 0.77 CCR2 (0.55) CCR2CYP3A4CYP2C9CYP2C19CCR4
SCHEMBL4904763 0.76 CCR2 (0.67) CCR2CYP3A4CYP2C9CYP2C19NFKBIA
SCHEMBL14006343 0.76 CCR2 (0.55) CCR2CYP3A4CYP2C9CYP2C19PIK3CA
SCHEMBL4904843 0.74 CCR2 (0.73) CCR2CYP3A4CYP2C9CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080293720-A1 Pyridinyl Sulfonamide Modulators of Chemokine Receptors GLAXO GROUP LIMITED (GB) 2008-11-27 US disclosed
US-20080293720-A1 Pyridinyl Sulfonamide Modulators of Chemokine Receptors GLAXO GROUP LIMITED (GB) 2008-11-27 US disclosed
US-20080293720-A1 Pyridinyl Sulfonamide Modulators of Chemokine Receptors GLAXO GROUP LIMITED (GB) 2008-11-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293720-A1 Pyridinyl Sulfonamide Modulators of Chemokine Receptors CCR2, CCR1, CCRL2 CCR2 1/4885PTGER4 343/4885PTGER2 77/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.