SCHEMBL4907620

SCHEMBL4907620

COc1ccc(COc2ccc([C@@](I)(CN)O[Si](C)(C)C(C)(C)C)c3ccc(=O)[nH]c23)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ADRB2 P07550 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ADRB1 P08588 1/20 0.33
CASP3 P42574 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
MAOB P27338 1/20 0.33
P2RY12 Q9H244 1/20 0.33
NTRK1 P04629 1/20 0.32
CSF1R P07333 1/20 0.32
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725393 0.79 ADRB2 (0.40) ARNPC1RAB9AADRB2MEN1
SCHEMBL17962298 0.75 APP (0.44) NPC1RAB9AADRB2MEN1KMT2A
SCHEMBL97964 0.72 MMP1 (0.44) NPC1RAB9AADRB2MEN1KMT2A
SCHEMBL2798225 0.70 MMP1 (0.41) NPC1RAB9AADRB2MEN1KMT2A
SCHEMBL19713174 0.68 ADRB2 (0.32) ADRB2ADRB1
SCHEMBL4786680 0.68 ADRB2 (0.41) ADRB2ADRB1MAOBMMP1MMP9
SCHEMBL19713173 0.68 ADRB2 (0.32) ADRB2ADRB1
SCHEMBL4786690 0.68 ADRB2 (0.41) ADRB2ADRB1MAOBMMP1MMP9
SCHEMBL14617522 0.68 ADRB2 (0.39) ADRB2ADRB1
SCHEMBL3586934 0.68 ADRB2 (0.39) ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008096129-A1 NITROGEN CONTAINING HETROCYCLIC COMPOUNDS USEFUL AS BIFUNCTIONAL MODULATORS OF M3 RECEPTORS AND BETA- 2 RECEPTORS ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed