SCHEMBL4908011

SCHEMBL4908011

Cc1cc(F)ccc1-c1cncc[n+]1[O-]

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 1/20 0.39
MAPK14 Q16539 5/20 0.37
GPBAR1 Q8TDU6 2/20 0.37
ALDH1A1 P00352 1/20 0.36
TDO2 P48775 1/20 0.36
NISCH Q9Y2I1 1/20 0.34
GRM5 P41594 1/20 0.34
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
PDE10A Q9Y233 2/20 0.33
HSP90AB1 P08238 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
TLR8 Q9NR97 1/20 0.32
PTGS2 P35354 1/20 0.32
ABL1 P00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4908287 0.74 MAPK14 (0.37) MAPK14ALDH1A1
SCHEMBL14164174 0.71 KCNA5 (0.38) KCNA5MAPK14GPBAR1ALDH1A1TDO2
SCHEMBL4897541 0.69
SCHEMBL4022519 0.68 NPC1 (0.48) KCNA5GPBAR1ALDH1A1TDO2GRM5
SCHEMBL16806032 0.68 TDO2 (0.54) KCNA5ALDH1A1TDO2GRM5CYP11B1
SCHEMBL26023290 0.68 HDAC8 (0.35) KCNA5MAPK14GRM5TLR8PTGS2
SCHEMBL14039912 0.68 PDE3B (0.44) KCNA5GPBAR1NISCHPDE10AHSP90AB1
SCHEMBL4902564 0.67 RAB9A (0.37) ALDH1A1NISCH
SCHEMBL12097254 0.67 GPBAR1 (0.47) KCNA5GPBAR1ALDH1A1TDO2GRM5
SCHEMBL26023434 0.67 GRIN2B (0.33) KCNA5GPBAR1TDO2GRM5GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed
US-20080132698-A1 Use of N-oxide compounds in coupling reactions UNIVERSITY OF OTTAWA 2008-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132698-A1 Use of N-oxide compounds in coupling reactions CYP4X1, CYP4F3, CYP1A2 KCNA5 1102/4885MAPK14 3470/4885GPBAR1 1164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.