Bromide

Bromide

SCHEMBL4908296

Br.C=CCc1ccccc1C(N)(CC=C)CC=C

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2B known ✓ P18089 2/20 0.30
ADRA2C known ✓ P18825 2/20 0.30
HTR1A known ✓ P08908 1/20 0.30
ADRA2A known ✓ P08913 1/20 0.30
GABRA1 P14867 2/20 0.38
GABRB2 P47870 2/20 0.38
HTT P42858 1/20 0.34
AKR1B1 P15121 1/20 0.33
ALDH1A1 P00352 3/20 0.33
TSHR P16473 1/20 0.33
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
VCAM1 P19320 1/20 0.32
KDM4E B2RXH2 1/20 0.31
IDO1 P14902 1/20 0.30
NISCH Q9Y2I1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL144630 0.98 GABRA1 (0.39) GABRA1GABRB2HTTAKR1B1ALDH1A1
Water SCHEMBL2836979 0.96 GABRA1 (0.38) GABRA1GABRB2HTTAKR1B1ALDH1A1
Hydrochloric Acid SCHEMBL668040 0.96 GABRA1 (0.38) GABRA1GABRB2HTTAKR1B1ALDH1A1
SCHEMBL10614506 0.83 GABRA1 (0.40) GABRA1GABRB2AKR1B1
SCHEMBL11667013 0.82 HTT (0.41) HTTALDH1A1TSHR
Hydrochloric Acid SCHEMBL10751108 0.81 GABRA1 (0.39) GABRA1GABRB2AKR1B1
SCHEMBL11056233 0.81 GABRA1 (0.41) GABRA1GABRB2HTTAKR1B1ALDH1A1
Bromide SCHEMBL9662608 0.80 GABRA1 (0.39) GABRA1GABRB2ALDH1A1TSHRICAM1
Iodide SCHEMBL19307326 0.79 GABRA1 (0.36) GABRA1GABRB2HTTALDH1A1TSHR
Hydrochloric Acid SCHEMBL11501232 0.78 GABRA1 (0.39) GABRA1GABRB2AKR1B1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994099-B1 Process for preparing 4-cyano-3-nitrobenzotrifluoride from 3-bromo-4-cyanobenzotrifluoride in the presence of catalytic cuprous cyanide and a phase transfer catalyst. BAYER CROPSCIENCE SA (FR) 2005-02-02 EP claimed
EP-1121344-A2 CHEMICAL PROCESSES AVENTIS CROPSCIENCE S.A. (FR) 2001-08-08 EP claimed
WO-2000021922-A2 CHEMICAL PROCESSES AVENTIS CROPSCIENCE S.A. (FR) 2000-04-20 WO claimed
EP-0994099-A1 Chemical processes Rhone Poulenc Agro (FR) 2000-04-19 EP claimed
US-4866183-A OXIDIZING TRIARYLIMIDAZOUS IN AQUEOUS ORGANIC TWO PHASE SYSTEM USING HYPOHALITE AND ONIUM SALT BASF AKTIENGESELLSCHAFT (DE) 1989-09-12 US claimed
US-3933768-A RUBBER BLENDS BRIDGESTONE TIRE COMPANY LIMITED (JA) 1976-01-20 US claimed
US-7364723-B1 Liquid preparation for contact lenses MENICON CO., LTD. (JP) 2008-04-29 US disclosed
EP-0994099-B1 Process for preparing 4-cyano-3-nitrobenzotrifluoride from 3-bromo-4-cyanobenzotrifluoride in the presence of catalytic cuprous cyanide and a phase transfer catalyst. BAYER CROPSCIENCE SA (FR) 2005-02-02 EP disclosed
EP-1214883-B1 LIQUID PREPARATION FOR CONTACT LENSES MENICON CO LTD (JP) 2003-11-26 EP disclosed
US-6635780-B1 For preparing intermediates of pesticides (particularly 4-cyano-3-nitrobenzotrifluoride); comprises the reaction of the corresponding ortho-nitrohalobenzene and metal cyanide, in a non aqueous solvent BAYER CROPSCIENCE S.A. (FR) 2003-10-21 US disclosed
EP-1214883-A1 LIQUID PREPARATION FOR CONTACT LENSES MENICON CO., LTD. (JP) 2002-06-19 EP disclosed
EP-1121344-A2 CHEMICAL PROCESSES AVENTIS CROPSCIENCE S.A. (FR) 2001-08-08 EP disclosed
WO-2000021922-A2 CHEMICAL PROCESSES AVENTIS CROPSCIENCE S.A. (FR) 2000-04-20 WO disclosed
EP-0994099-A1 Chemical processes Rhone Poulenc Agro (FR) 2000-04-19 EP disclosed
US-3933768-A RUBBER BLENDS BRIDGESTONE TIRE COMPANY LIMITED (JA) 1976-01-20 US disclosed