SCHEMBL491077

SCHEMBL491077

CCOC(=O)CCc1cc(OC)c(OC)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
KMT2A Q03164 7/20 0.59
MEN1 O00255 2/20 0.59
KDM4E B2RXH2 1/20 0.59
MAPT P10636 2/20 0.56
GAA P10253 2/20 0.54
CYP4F2 P78329 1/20 0.53
CYP4A11 Q02928 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3492958 0.90 ALDH1A1 (0.53) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL490309 0.87 ALOX5 (0.66) ALDH1A1KMT2AGAACYP4F2CYP4A11
SCHEMBL28222447 0.85 KMT2A (0.55) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL7431362 0.85 MAPT (0.63) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL3457181 0.83 ALDH1A1 (0.70) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL491276 0.83 CYP4F2 (0.59) KMT2AMEN1KDM4ECYP4F2CYP4A11
SCHEMBL12812251 0.82 KMT2A (0.51) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL8912630 0.81 CYP4F2 (0.58) ALDH1A1KMT2ACYP4F2CYP4A11
SCHEMBL9832305 0.81 ALDH1A1 (0.56) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL11212268 0.81 ALOX5 (0.55) ALDH1A1KMT2ACYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2994460-B1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES UNIV INDIANA RES & TECH CORP (US) 2024-12-04 EP disclosed
US-10738024-B2 Compounds for treatment of angiogenesis-mediated diseases INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2020-08-11 US disclosed
US-10238627-B2 Compounds for treatment of angiogenesis-mediated diseases INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2019-03-26 US disclosed
US-20180177758-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION 2018-06-28 US disclosed
EP-2994460-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES Indiana University Research and Technology Corporation (US) 2016-03-16 EP disclosed
US-20160060241-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES GACHON UNIVERSITY OF INDUSTRY-ACADEMIC COOPERATION FOUNDATION (KR) 2016-03-03 US disclosed
WO-2014182695-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION (US) 2014-11-13 WO disclosed
US-8268293-B2 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2012-09-18 US disclosed
CN-101163659-B Antioxidants MERCK PATENT GMBH 2012-09-05 CN disclosed
US-8106233-B2 Applying di-2-ethylhexyl 4-hydroxy-3,5-dimethoxy-benzylmalonate; protective action against UV rays, oxidative stress on body cells, counters skin ageing MERCK PATENT GMBH (DE) 2012-01-31 US disclosed
US-5414108-A From a Meldrum's acid derivative BIOGAL GYOGYSZERGRAR (HU) 1995-05-09 US disclosed
US-5350872-A Decyclization and decarboxylation of a 1,3-dioxane-4,6-dione BIOGAL GYOGYSZERGRAR (HU) 1994-09-27 US disclosed
EP-0578850-A1 Process for the preparation of carboxylic acids and derivatives of them BIOGAL GYOGYSZERGYAR (HU) 1994-01-19 EP disclosed
US-4523015-A Process and nitroaminopyrimidone intermediates for histamine H2 -antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-06-11 US disclosed
EP-0004793-B1 2-NITRO AMINOPYRIMIDONE DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND THEIR USE TO PREPARE 2-AMINOPYRIMIDONE DERIVATIVES WHICH HAVE HISTAMINE H2-ANTAGONIST ACTIVITY SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1981-12-30 EP disclosed
US-4227000-A Intermediates in the process for making histamine antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-10-07 US disclosed
US-4218452-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-08-19 US disclosed
EP-0004793-A2 2-nitro aminopyrimidone derivatives, a process for their preparation and their use to prepare 2-aminopyrimidone derivatives which have histamine H2-antagonist activity SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-10-17 EP disclosed
US-4159329-A BLOCKING AGENTS, ANTAGONISTS, ANTIHISTAMINES SMITHKLINE & FRENCH LABORATORIES LIMITED (GB) 1979-06-26 US disclosed
US-4145546-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-03-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10738024-B2 Compounds for treatment of angiogenesis-mediated diseases KDR, TEK, VEGFA ALDH1A1 1077/4885KMT2A 4465/4885MEN1 2818/4885
US-20180177758-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES KDR, TEK, VEGFA ALDH1A1 1077/4885KMT2A 4465/4885MEN1 2818/4885
US-20160060241-A1 COMPOUNDS FOR TREATMENT OF ANGIOGENESIS-MEDIATED DISEASES KDR, TEK, VEGFA ALDH1A1 1077/4885KMT2A 4465/4885MEN1 2818/4885
US-10238627-B2 Compounds for treatment of angiogenesis-mediated diseases KDR, TEK, VEGFA ALDH1A1 1077/4885KMT2A 4465/4885MEN1 2818/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.