SCHEMBL4923969

SCHEMBL4923969

CC(C)(C)OC(=O)N1C[C@H](OS(C)(=O)=O)C[C@H]1C(=O)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 7/20 0.45
ABCB1 P08183 1/20 0.44
KLK7 P49862 1/20 0.43
FKBP1A P62942 3/20 0.42
NR1H2 P55055 2/20 0.42
NR1H3 Q13133 2/20 0.42
GPR119 Q8TDV5 2/20 0.41
UCHL1 P09936 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1781450 1.00 MCL1 (0.45) MCL1ABCB1KLK7FKBP1ANR1H2
SCHEMBL1781452 1.00 MCL1 (0.45) MCL1ABCB1KLK7FKBP1ANR1H2
SCHEMBL7149261 0.92 POLB (0.43) MCL1ABCB1KLK7POLB
SCHEMBL21066263 0.91 KLK7 (0.47) MCL1ABCB1KLK7FKBP1ANR1H2
SCHEMBL22322657 0.90 KLK7 (0.48) KLK7FKBP1ANR1H2NR1H3
SCHEMBL29550939 0.90 KLK7 (0.48) KLK7FKBP1ANR1H2NR1H3
SCHEMBL1448111 0.87 ABCB1 (0.54) MCL1ABCB1KLK7FKBP1AUCHL1
SCHEMBL21273903 0.87 ABCB1 (0.54) MCL1ABCB1KLK7FKBP1AUCHL1
SCHEMBL7703700 0.87 ABCB1 (0.54) MCL1ABCB1KLK7FKBP1AUCHL1
SCHEMBL7279798 0.87 ABCB1 (0.54) MCL1ABCB1KLK7FKBP1AUCHL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4678238-A2 ARGINASE INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2026-01-14 EP disclosed
US-20250313578-A1 Arginase Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2025-10-09 US disclosed
EP-3752251-B1 ARGINASE INHIBITORS AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2025-09-10 EP disclosed
US-12195485-B2 Arginase inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2025-01-14 US disclosed
US-11912727-B2 Arginase inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2024-02-27 US disclosed
CN-117180290-A Arginase inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2023-12-08 CN disclosed
US-20230365599-A1 Arginase Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2023-11-16 US disclosed
CN-111712302-B Arginase inhibitors and methods of use thereof 阿斯利康(瑞典)有限公司 2023-09-19 CN disclosed
US-20230122859-A1 Arginase Inhibitors and Methods of Use Thereof ASTRAZENECA AB (SE) 2023-04-20 US disclosed
US-11420984-B2 Arginase inhibitors and methods of use thereof ASTRAZENECA AB (SE) 2022-08-23 US disclosed
US-20080119464-A1 PHARMACEUTICAL COMPOSITIONS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) ABBVIE INC. 2008-05-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11912727-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 MCL1 1172/4885ABCB1 870/4885KLK7 4255/4885
US-12195485-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, PRMT1 MCL1 905/4885ABCB1 815/4885KLK7 4347/4885
US-20230122859-A1 Arginase Inhibitors and Methods of Use Thereof ARG1, ARG2, PRMT1 MCL1 905/4885ABCB1 815/4885KLK7 4347/4885
US-20080119464-A1 PHARMACEUTICAL COMPOSITIONS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) DPP4, DPP3, DPP7 MCL1 3879/4885ABCB1 329/4885KLK7 1127/4885
US-20230365599-A1 Arginase Inhibitors and Methods of Use Thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 MCL1 1172/4885ABCB1 870/4885KLK7 4255/4885
US-20250313578-A1 Arginase Inhibitors and Methods of Use Thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 MCL1 1172/4885ABCB1 870/4885KLK7 4255/4885
US-11420984-B2 Arginase inhibitors and methods of use thereof ARG1, ARG2, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 MCL1 1110/4885ABCB1 863/4885KLK7 4247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.