SCHEMBL4934640

SCHEMBL4934640

Cc1c(F)cc(-c2ccc(O)cc2)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SENP1 Q9P0U3 1/20 0.42
ESR1 P03372 10/20 0.41
APP P05067 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
RPS6KA3 P51812 2/20 0.40
ESR2 Q92731 6/20 0.40
ABL1 P00519 1/20 0.39
ABCB1 P08183 1/20 0.39
BCR P11274 1/20 0.39
KIF11 P52732 1/20 0.39
USP7 Q93009 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320686 0.83 PTGS2 (0.50) RPS6KA3
SCHEMBL27639098 0.82 USP7 (0.46) ESR1APPCYP3A4CYP2C9CYP2C19
SCHEMBL16982131 0.82 RPS6KA3 (0.49) SENP1ESR1RPS6KA3ESR2ABL1
SCHEMBL7077947 0.79 DHODH (0.40) CYP2C9CYP2C19RPS6KA3ESR2
SCHEMBL27928527 0.78 ESR1 (0.57) ESR1APPCYP3A4CYP2C9CYP2C19
SCHEMBL27639192 0.78 ESR1 (0.41) ESR1APPCYP3A4CYP2C9CYP2C19
SCHEMBL25420748 0.78 RPS6KA3 (0.49) SENP1ESR1RPS6KA3ESR2ABL1
SCHEMBL1759436 0.78 ESR2 (0.47) ESR1APPCYP3A4CYP2C9CYP2C19
SCHEMBL9318422 0.77 GCGR (0.38)
SCHEMBL13105050 0.77 ESR1 (0.56) SENP1ESR1ESR2ABL1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7329777-B2 Methods for treating heart failure, thromboembolic disorders, and pulmonary fibrosis BAYER AKTIENGESELLSCHAFT (DE) 2008-02-12 US disclosed
US-6939990-B2 Derivatives of dicarboxylic acid having pharmaceutical properties BAYER AKTIENGESELLSCHAFT (DE) 2005-09-06 US disclosed