SCHEMBL4942622

SCHEMBL4942622

CC(C)c1cc2c(=O)c(C#N)c[nH]c2s1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.35
DPYD Q12882 1/20 0.33
KDM5A P29375 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3997496 0.80 DPYD (0.36) MCL1DPYDKDM5A
SCHEMBL3996464 0.77 TMIGD3 (0.39) DPYDKDM5A
SCHEMBL3993861 0.71 KDM4E (0.46) MCL1
SCHEMBL3995033 0.69 HPGD (0.39) MCL1
SCHEMBL3999236 0.69 KDM5A (0.34) MCL1DPYDKDM5A
SCHEMBL3997640 0.67 DPYD (0.38) MCL1DPYD
SCHEMBL15850393 0.66 IMPDH2 (0.39) MCL1DPYD
SCHEMBL18332827 0.65 DPYD (0.43) MCL1DPYDKDM5A
SCHEMBL3999985 0.65 DPYD (0.36) MCL1DPYD
SCHEMBL4847045 0.62 GRM6 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937690-A1 THIENO[2,3-B]PYRIDINE-5-CARBONITRILES AS PROTEIN KINASE INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2008-07-02 EP disclosed
WO-2007038519-A1 THIENO[2,3-B]PYRIDINE-5-CARBONITRILES AS PROTEIN KINASE INHIBITORS WYETH (US) 2007-04-05 WO disclosed