SCHEMBL4948159

SCHEMBL4948159

N#Cc1ccccc1-c1ccc(-c2sccc2N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.51
PTPN5 P54829 1/20 0.41
PTGS1 P23219 1/20 0.41
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
TRPA1 O75762 1/20 0.38
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 3/20 0.36
CLK4 Q9HAZ1 2/20 0.36
MAPK1 P28482 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
GRM6 O15303 1/20 0.36
PRKAG1 P54619 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4953419 0.82 PTGS1 (0.39) ESR2PTGS1ALOX5APFEN1CYP1A2
SCHEMBL4950501 0.82 PTGS1 (0.39) ESR2PTGS1CYP1A2CYP3A4ALDH1A1
SCHEMBL4948327 0.81 STS (0.49) ESR2PTGS1ALDH1A1CLK4
SCHEMBL4948367 0.80 ESR2 (0.43) ESR2PTGS1MEN1KMT2APTGS2
SCHEMBL4950454 0.80 PTGS1 (0.50) PTGS1GABRG2GABRB3GABRA5GABRA3
SCHEMBL4948155 0.80 ESR2 (0.50) ESR2PTPN5PTGS1ALDH1A1MAPK1
SCHEMBL4359377 0.76 ESR2 (0.66) ESR2PTPN5ALOX5APFEN1TRPA1
SCHEMBL8382823 0.76 ESR2 (0.47) ESR2PTPN5PTGS1CYP1A2ALDH1A1
SCHEMBL31410710 0.75 ESR2 (0.76) ESR2PTPN5ALOX5APFEN1TRPA1
SCHEMBL4950460 0.74 VCAM1 (0.42) CYP3A4ALDH1A1MEN1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893597-B1 AMPA RECEPTOR POTENTIATORS LILLY CO ELI (US) 2008-11-12 EP disclosed