SCHEMBL4948557

SCHEMBL4948557

COc1cc(C(=O)C2=C(C(F)(F)F)N=CCC2=O)cc([N+](=O)[O-])c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 3/20 0.51
FTO Q9C0B1 1/20 0.39
LMNA P02545 2/20 0.37
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EGFR P00533 1/20 0.36
POLB P06746 2/20 0.36
JUN P05412 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GAA P10253 2/20 0.35
RAB9A P51151 1/20 0.35
GFER P55789 1/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4943343 0.86 TTR (0.53) TTRFTOLMNAMAPTTDP1
SCHEMBL7371244 0.73 TTR (0.71) TTRLMNAMAPTSMN1; SMN2POLB
SCHEMBL7367724 0.70 TTR (0.57) TTRLMNAMAPTJUNTDP1
SCHEMBL3584563 0.69 TTR (0.53) TTRFTOLMNAMAPTPOLB
SCHEMBL7369924 0.69 TTR (0.64) TTRFTOLMNAMAPTSMN1; SMN2
SCHEMBL7365333 0.69 TTR (0.75) TTRLMNAMAPTSMN1; SMN2EGFR
SCHEMBL3583434 0.69 CA12 (0.66) TTRFTOMAPTSMN1; SMN2EGFR
SCHEMBL5598228 0.69 LMNA (0.66) TTRFTOLMNAMAPTSMN1; SMN2
SCHEMBL31059024 0.69 LMNA (0.66) TTRFTOLMNAMAPTSMN1; SMN2
SCHEMBL31059025 0.69 LMNA (0.66) TTRFTOLMNAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed