SCHEMBL4948715

SCHEMBL4948715

CC(C)(C)OC(=O)OC(=O)CCCCCNS(=O)(=O)c1ccc(Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.56
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.46
PKM P14618 2/20 0.46
HTT P42858 1/20 0.46
TBXA2R P21731 1/20 0.45
LMNA P02545 2/20 0.45
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19450350 0.86 GAA (0.54) ALDH1A1GAAPKMTBXA2RLMNA
SCHEMBL15797966 0.83 ALDH1A1 (0.65) ALDH1A1GAATSHRPKMHTT
SCHEMBL6670344 0.82 ALDH1A1 (0.62) ALDH1A1GAATSHRPKMHTT
SCHEMBL4950063 0.82 ALDH1A1 (0.61) ALDH1A1GAATSHRPKMHTT
SCHEMBL24762017 0.81 ALDH1A1 (0.60) ALDH1A1GAATSHRPKM
SCHEMBL19450347 0.80 SIGMAR1 (0.50) ALDH1A1GAASIGMAR1
SCHEMBL7945710 0.78 ALDH1A1 (0.64) ALDH1A1GAAPKMLMNASIGMAR1
SCHEMBL17680506 0.77 ALDH1A1 (0.55) ALDH1A1GAATSHRSIGMAR1
SCHEMBL931443 0.77 ALDH1A1 (0.50) ALDH1A1TSHRPKMHTTTBXA2R
SCHEMBL9870160 0.76 ALDH1A1 (0.75) ALDH1A1TSHRPKMTBXA2RLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1921062-A2 Amino acid derivatives as HIV aspartyl protease inhibitors Ambrilia Biopharma Inc. (CA) 2008-05-14 EP disclosed
US-20060079550-A1 Amino acid derivatives useful for the treatment of alzheimer's disease ELAN PHARMACEUTICALS, INC. 2006-04-13 US disclosed
EP-1263716-A2 AMINO ACID DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS Pharmacor Inc. (CA) 2002-12-11 EP disclosed
US-6455587-B1 AROMATIC SULFONYL DERIVATIVES PHARMACOR INC. (CA) 2002-09-24 US disclosed
WO-2001068593-A2 AMINO ACID DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS PHARMACOR INC. (CA) 2001-09-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079550-A1 Amino acid derivatives useful for the treatment of alzheimer's disease BACE1, APP, PSEN1 ALDH1A1 2554/4885GAA 197/4885TSHR 3263/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.