SCHEMBL4948719

SCHEMBL4948719

N#C/C(=C/c1c(Cl)cncc1Cl)c1cc(O)c(O)c([N+](=O)[O-])c1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 8/20 0.61
COMT P21964 4/20 0.50
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
RECQL P46063 1/20 0.47
KMT2A Q03164 1/20 0.47
TTR P02766 1/20 0.45
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3589543 0.79 FTO (0.71) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL3589548 0.79 FTO (0.71) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL4946977 0.76 FTO (0.47) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL4943899 0.76 FTO (0.47) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL20100844 0.76 FTO (1.00) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL29493661 0.75 FTO (0.53) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL3586620 0.75 TTR (0.65) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL4948407 0.74 COMT (0.46) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL4948470 0.72 FTO (0.45) FTOCOMTMEN1ALDH1A1MAPT
SCHEMBL20100839 0.71 FTO (1.00) FTOCOMTMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed