SCHEMBL4948734

SCHEMBL4948734

Cc1cc(S(=O)(=O)c2cccc(C(=O)N(C)C)c2)c2ncc(C(N)=O)c(Nc3ccc4ncn(C)c4c3)c2c1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 19/20 0.54
PDE4A P27815 2/20 0.45
PDE4C Q08493 2/20 0.45
PDE4D Q08499 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2478457 0.89 PDE4B (0.58) PDE4BPDE4APDE4CPDE4D
SCHEMBL4946623 0.83 PDE4B (0.73) PDE4BPDE4APDE4CPDE4D
SCHEMBL4948833 0.81 PDE4B (0.52) PDE4B
SCHEMBL4946650 0.76 PDE4B (0.56) PDE4BPDE4APDE4CPDE4D
SCHEMBL1276426 0.75 PDE4B (0.72) PDE4B
SCHEMBL4950488 0.75 PDE4B (0.50) PDE4BPDE4APDE4CPDE4D
SCHEMBL4948174 0.74 PDE4B (0.76) PDE4BPDE4APDE4CPDE4D
SCHEMBL2481933 0.74 PDE4B (0.64) PDE4BPDE4APDE4CPDE4D
SCHEMBL4944370 0.73 PDE4B (0.38) PDE4B
SCHEMBL4952284 0.72 PDE4B (0.45) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed