SCHEMBL4948740

SCHEMBL4948740

O=C1CC=NC(C(F)(F)F)=C1c1nccc(-c2cc(O)c(O)c([N+](=O)[O-])c2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 5/20 0.37
KDM4E B2RXH2 4/20 0.34
MEN1 O00255 4/20 0.34
ALDH1A1 P00352 4/20 0.34
MAPT P10636 4/20 0.34
KMT2A Q03164 4/20 0.34
RECQL P46063 3/20 0.34
TDP1 Q9NUW8 3/20 0.34
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
LMNA P02545 2/20 0.34
THRB P10828 2/20 0.34
BLM P54132 2/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
CASP6 P55212 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAOA P21397 3/20 0.33
MAOB P27338 2/20 0.33
CRHBP P24387 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948714 0.83 MAPT (0.37) MEN1ALDH1A1MAPTKMT2ALMNA
SCHEMBL1447172 0.82 COMT (0.46) TTRMAPTPOLBGAATP53
SCHEMBL4951393 0.78 TTR (0.34) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3585312 0.75 TTR (0.41) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL4949041 0.74 TTR (0.35) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3595074 0.73 MAPT (0.44) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3588381 0.73 TTR (0.45) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3587064 0.73 TTR (0.39) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3591192 0.73 TTR (0.39) TTRKDM4EMEN1ALDH1A1MAPT
SCHEMBL3586419 0.72 MAPT (0.39) TTRKDM4EMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed