SCHEMBL4948827

SCHEMBL4948827

CCc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3ccc(F)c(OC)c3)c2c1

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.71
CSF1R P07333 16/20 0.55
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4951386 0.89 PDE4B (0.74) PDE4BCSF1R
SCHEMBL4950158 0.86 PDE4B (0.73) PDE4BCSF1R
SCHEMBL2475119 0.85 PDE4B (0.83) PDE4BCSF1R
SCHEMBL4948930 0.84 CSF1R (0.53) PDE4BCSF1R
SCHEMBL1275852 0.81 PDE4B (1.00) PDE4BCSF1R
SCHEMBL1275858 0.81 PDE4B (0.85) PDE4BCSF1R
SCHEMBL4949284 0.79 PDE4B (0.60) PDE4BCSF1R
SCHEMBL4949687 0.79 PDE4B (0.44) PDE4BCSF1R
SCHEMBL4952317 0.78 PDE4B (0.68) PDE4BCSF1R
SCHEMBL12115499 0.78 PDE4B (0.78) PDE4BCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed