SCHEMBL4948930

SCHEMBL4948930

CCc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3cccc(F)c3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 6/20 0.53
PDE4B Q07343 13/20 0.50
LMNA P02545 1/20 0.45
LRRK2 Q5S007 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949063 0.88 CSF1R (0.56) CSF1RPDE4BLMNALRRK2
SCHEMBL4948831 0.88 PDE4B (0.56) CSF1RPDE4BLMNALRRK2
SCHEMBL4952317 0.86 PDE4B (0.68) CSF1RPDE4B
SCHEMBL4949284 0.86 PDE4B (0.60) CSF1RPDE4BLRRK2
SCHEMBL2479835 0.84 PDE4B (0.60) CSF1RPDE4BLRRK2
SCHEMBL4948827 0.84 PDE4B (0.71) CSF1RPDE4B
SCHEMBL4949687 0.80 PDE4B (0.44) CSF1RPDE4BLRRK2
SCHEMBL1276135 0.80 PDE4B (0.75) CSF1RPDE4BLRRK2
SCHEMBL27670097 0.80 CSF1R (0.53) CSF1RPDE4BLMNA
SCHEMBL1275872 0.79 PDE4B (0.61) CSF1RPDE4BLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed