SCHEMBL4948857

SCHEMBL4948857

COC(=O)c1ccc(C#C[C@@]2(O)CCCN2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PKM P14618 1/20 0.38
GRM5 P41594 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HPGD P15428 1/20 0.37
PTPN11 Q06124 1/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 1/20 0.36
NR1H2 P55055 1/20 0.35
GRM3 Q14832 1/20 0.35
JAK3 P52333 1/20 0.35
KDM4E B2RXH2 1/20 0.35
XBP1 P17861 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23883988 0.80 PKM (0.44) HDAC1HDAC6PKMGRM5SMN1; SMN2
SCHEMBL23900037 0.80 PKM (0.44) HDAC1HDAC6PKMGRM5SMN1; SMN2
SCHEMBL23899816 0.75 PTPN11 (0.42) HDAC1HDAC6PKMPTPN11JAK2
SCHEMBL28516359 0.74 ALDH1A1 (0.52) GRM5SMN1; SMN2HPGDPTPN11MAPT
SCHEMBL27363769 0.74 ALDH1A1 (0.55) GRM5SMN1; SMN2HPGDPTPN11NPC1
SCHEMBL25427135 0.74 HDAC1 (0.42) HDAC1HDAC6PKMSMN1; SMN2HPGD
SCHEMBL25427129 0.74 HDAC1 (0.42) HDAC1HDAC6PKMSMN1; SMN2HPGD
SCHEMBL5155331 0.74 MAPT (0.43) HDAC1HDAC6PKMSMN1; SMN2NPC1
SCHEMBL27363966 0.73 ALDH1A1 (0.57) GRM5SMN1; SMN2HPGDPTPN11NPC1
SCHEMBL31386140 0.70 PKM (0.44) HDAC1HDAC6PKMSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed
EP-1961750-A1 VLA-4 INHIBITORY DRUG Daiichi Sankyo Company, Limited (JP) 2008-08-27 EP disclosed