SCHEMBL4949150

SCHEMBL4949150

CCOc1cccc(S(=O)(=O)c2cc(C)cc3c(Nc4cccc(OC)c4)c(C(N)=O)cnc23)c1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 18/20 0.64
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
PDE4A P27815 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
CSF1R P07333 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4946547 0.91 PDE4B (0.77) PDE4BPDE4APDE4CPDE4D
SCHEMBL4948739 0.89 PDE4B (0.71) PDE4BPDE4APDE4CPDE4DCSF1R
SCHEMBL4944841 0.89 PDE4B (0.77) PDE4BPDE4APDE4CPDE4DCSF1R
SCHEMBL4952294 0.89 PDE4B (0.66) PDE4BPDE4APDE4CPDE4DCSF1R
SCHEMBL1276415 0.88 PDE4B (0.83) PDE4BTP53MAPTPDE4APDE4C
SCHEMBL4946623 0.87 PDE4B (0.73) PDE4BPDE4APDE4CPDE4D
SCHEMBL4946407 0.82 PDE4B (0.66) PDE4BCSF1R
SCHEMBL4949236 0.82 PDE4B (0.66) PDE4BCSF1R
SCHEMBL4952552 0.81 PDE4B (0.65) PDE4BTP53CSF1R
SCHEMBL4949011 0.81 PDE4B (0.58) PDE4BTP53MAPTPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed