Normetanephrine

Normetanephrine

SCHEMBL4949341

COc1cc([C@@H](O)CN)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 1.00
BLM P54132 6/20 0.97
PMP22 Q01453 3/20 0.97
TSHR P16473 4/20 0.73
CYP3A4 P08684 2/20 0.73
SLC22A3 O75751 1/20 0.63
MAPT P10636 3/20 0.62
RECQL P46063 3/20 0.62
TDP1 Q9NUW8 3/20 0.62
TAAR1 Q96RJ0 3/20 0.62
MAPK1 P28482 3/20 0.62
LMNA P02545 3/20 0.62
KDM4E B2RXH2 3/20 0.62
HPGD P15428 2/20 0.62
APEX1 P27695 2/20 0.62
ADRA2A P08913 2/20 0.62
ADRA1A P35348 2/20 0.62
MEN1 O00255 1/20 0.62
ADRB2 P07550 1/20 0.62
ADRB1 P08588 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Normetanephrine SCHEMBL137755 1.00 NFKB1 (1.00) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine SCHEMBL29516838 1.00 NFKB1 (1.00) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine SCHEMBL1168235 0.98 BLM (1.00) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine SCHEMBL15421560 0.97 NFKB1 (0.94) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine SCHEMBL11341275 0.92 NFKB1 (0.85) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine SCHEMBL28288010 0.91 NFKB1 (0.83) NFKB1BLMPMP22TSHRCYP3A4
Metanephrine SCHEMBL2771744 0.90 NFKB1 (0.81) NFKB1BLMPMP22TSHRCYP3A4
SCHEMBL3175780 0.86 NFKB1 (0.74) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine Hydrochloride SCHEMBL7153624 0.86 NFKB1 (0.76) NFKB1BLMPMP22TSHRCYP3A4
Normetanephrine Hydrochloride SCHEMBL11573078 0.86 NFKB1 (0.76) NFKB1BLMPMP22TSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4181781-B1 BREATH-BASED THERAPEUTIC DRUG MONITORING METHOD UNIV KINDERSPITAL BEIDER BASEL (CH) 2026-05-20 EP disclosed
US-20250044306-A1 Methods for Determining Opioid Responsiveness in the Treatment of Pain EAST CAROLINA UNIVERSITY 2025-02-06 US disclosed
US-20230277125-A1 BREATH-BASED THERAPEUTIC DRUG MONITORING METHOD UNIVERSITÄTS-KINDERSPITAL BEIDER BASEL (CH) 2023-09-07 US disclosed
WO-2023028350-A1 THERAPEUTIC COMPOSITIONS AND RELATED METHODS BOYCE THOMPSON INSTITUTE FOR PLANT RESEARCH, INC. (US) 2023-03-02 WO disclosed
US-20080167318-A1 Pharmaceutically active pyrrolidine derivatives APPLIED RESEARCH SYSTEM ARS HOLDING N.V. (NL) 2008-07-10 US disclosed
US-7211601-B2 Pharmaceutically active pyrrolidine derivatives APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2007-05-01 US disclosed
EP-1268419-B1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-21 EP disclosed
EP-1268418-B1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS (AN) 2006-06-14 EP disclosed
US-7018988-B2 Pharmaceutically active pyrrolidine derivatives as Bax inhibitors APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2006-03-28 US disclosed
US-20030212012-A1 Pharmaceutically active pyrrolidine derivatives MERCK SERONO SA (CH) 2003-11-13 US disclosed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed
US-6114582-A DECYCLIZATION TO FORM A CHEMICAL INTERMEDIATE FOR PRODUCING AN ANTI-OBESITY AGENT AND ANTIDIABETIC AGENT DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-05 US disclosed
EP-0654534-B1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEM (JP) 2000-03-01 EP disclosed
EP-0939134-A1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-09-01 EP disclosed
EP-0924194-A2 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-06-23 EP disclosed
EP-0924193-A1 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1999-06-23 EP disclosed
US-5811293-A CULTURE PRODUCT AS CHEMICAL INTERMEDIATE FOR ANTI-OBESITY AGENT DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-22 US disclosed
US-5629200-A MICROORGANISM DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-13 US disclosed
EP-0654534-A2 Processes for producing optically active 2-amino-1-phenylethanol derivatives DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030212012-A1 Pharmaceutically active pyrrolidine derivatives OXTR, CNR1, PRLHR NFKB1 1472/4885BLM 4611/4885PMP22 1055/4885
US-20080167318-A1 Pharmaceutically active pyrrolidine derivatives OXTR, PRLHR, NR0B1 NFKB1 1588/4885BLM 4441/4885PMP22 1567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.