SCHEMBL4949949

SCHEMBL4949949

N#Cc1ccccc1-c1ccc(-c2ccncc2N)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.51
PDE10A Q9Y233 1/20 0.50
ALOX5AP P20292 1/20 0.44
FEN1 P39748 1/20 0.44
TRPA1 O75762 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20189792 0.80 CYP11B2 (0.51) GSK3AGSK3B
SCHEMBL3224025 0.79 ESR2 (0.60) ESR2PDE10ATRPA1GSK3AGSK3B
SCHEMBL31663514 0.79 ESR2 (0.60) ESR2PDE10ATRPA1GSK3AGSK3B
SCHEMBL28162273 0.79 CYP1A2 (0.45) ESR2PDE10AALOX5APFEN1CYP1A2
SCHEMBL13316726 0.78 HTT (0.50) ESR2PDE10ATRPA1CYP1A2CYP3A4
SCHEMBL3791281 0.77 ALDH1A1 (0.54) GSK3BCYP1A2CYP3A4CYP2C19CYP2E1
SCHEMBL1146097 0.76 CYP1A2 (0.57) ESR2PDE10ACYP1A2CYP3A4CYP2C19
SCHEMBL7215513 0.76 ATR (0.50) ESR2PDE10ACYP1A2CYP3A4CYP2C19
SCHEMBL4359377 0.76 ESR2 (0.66) ESR2PDE10AALOX5APFEN1TRPA1
Hydrochloric Acid SCHEMBL16702548 0.76 ALDH1A1 (0.52) GSK3BCYP1A2CYP3A4CYP2C19CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893597-B1 AMPA RECEPTOR POTENTIATORS LILLY CO ELI (US) 2008-11-12 EP disclosed