SCHEMBL4950023

SCHEMBL4950023

Cc1c(O)cc2c(c1Cl)C(=O)C(C1CCCC1)C2

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.39
ADRB3 P13945 1/20 0.38
GPR183 P32249 1/20 0.38
ACHE P22303 2/20 0.32
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
ATM Q13315 1/20 0.31
ACLY P53396 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4941945 0.87 GRM2 (0.44) GRM2ADRB3GPR183ACHEMAPT
SCHEMBL4945422 0.87 GRM2 (0.43) GRM2ADRB3GPR183ACHEACLY
SCHEMBL11654170 0.81 GRM2 (0.44) GRM2ADRB3GPR183ACHEMAPT
SCHEMBL11027295 0.74 GRM2 (0.50) GRM2ADRB3GPR183ACHEMAPT
SCHEMBL11659608 0.74 GRM2 (0.41) GRM2ADRB3GPR183ACHE
SCHEMBL11708448 0.74 MAPT (0.34) GRM2MAPT
SCHEMBL11708654 0.74 NPC1 (0.38) GRM2ADRB3GPR183MAPT
SCHEMBL11707808 0.72 LMNA (0.35) GRM2MAPT
SCHEMBL11654377 0.70 GRM2 (0.50) GRM2ADRB3GPR183ACHEMAPT
SCHEMBL22804010 0.69 GRM2 (0.52) GRM2ADRB3GPR183MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080312286-A1 Indanone Potentiators of Metabotropic Glutamate Receptors MERCK SHARP & DOHME CORP. 2008-12-18 US disclosed
EP-1773792-A1 INDANONE POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS Merck & Co., Inc. (US) 2007-04-18 EP disclosed
WO-2006015158-A1 INDANONE POTENTIATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080312286-A1 Indanone Potentiators of Metabotropic Glutamate Receptors GRM2, GRIK2, GRM1 GRM2 1/4885ADRB3 708/4885GPR183 186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.