SCHEMBL4950026

SCHEMBL4950026

CC(NC(=O)C(O)c1ccc(C(F)(F)F)cc1)C(=O)Nc1cc(C(C)Cc2ccccc2)nn1C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ6 P48051 2/20 0.39
KCNJ5 P48544 2/20 0.39
KCNJ3 P48549 2/20 0.39
LDHB P07195 1/20 0.38
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
POLB P06746 2/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
CNR2 P34972 1/20 0.37
FPR2 P25090 1/20 0.37
PKM P14618 1/20 0.36
CTSL P07711 1/20 0.36
CTSK P43235 1/20 0.36
PDE2A O00408 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949144 0.92 PSMB5 (0.39) POLBMAPTPKM
SCHEMBL4958532 0.90 MMP1 (0.38) KCNJ6KCNJ5KCNJ3MMP1MMP2
SCHEMBL4950030 0.85 EP300 (0.37) LDHBMMP1MMP2MMP9MMP8
SCHEMBL8320609 0.82 MAPK13 (0.39) KCNJ6KCNJ5KCNJ3LDHBMMP1
SCHEMBL2954505 0.82 MAPK13 (0.39) KCNJ6KCNJ5KCNJ3LDHBMMP1
SCHEMBL4948937 0.79 PSMB5 (0.37) POLBPKM
SCHEMBL4949147 0.77 POLB (0.39) POLBPKM
SCHEMBL4946819 0.77 PSEN1 (0.44)
SCHEMBL4948096 0.75 PSEN1 (0.41) POLBCNR2PKM
SCHEMBL4958535 0.75 MALT1 (0.39) MMP1MMP2MMP9MMP8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633350-A4 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARM INC (US) 2008-11-26 EP disclosed
EP-1633350-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2006-03-15 EP disclosed
WO-2005009344-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 2005-02-03 WO disclosed