SCHEMBL4958532

SCHEMBL4958532

CC(NC(=O)C(O)c1ccc(Cl)cc1)C(=O)Nc1cc(C(C)Cc2ccccc2)nn1C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.38
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP8 P22894 2/20 0.38
CNR1 P21554 5/20 0.36
KCNJ6 P48051 1/20 0.36
KCNJ5 P48544 1/20 0.36
KCNJ3 P48549 1/20 0.36
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
CYP2C19 P33261 1/20 0.35
MALT1 Q9UDY8 1/20 0.35
ATM Q13315 1/20 0.35
PDE1C Q14123 2/20 0.35
SDCBP O00560 1/20 0.35
SDC2 P34741 1/20 0.35
CNR2 P34972 4/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949144 0.94 PSMB5 (0.39) POLBPKMATMMEN1KMT2A
SCHEMBL4950026 0.90 KCNJ6 (0.39) MMP1MMP2MMP9MMP8KCNJ6
SCHEMBL4958535 0.85 MALT1 (0.39) MMP1MMP2MMP9MMP8CNR1
SCHEMBL2965613 0.81 MAPK14 (0.40) POLBPKMCYP3A4GAACYP2C19
SCHEMBL8318851 0.81 MAPK14 (0.40) POLBPKMCYP3A4GAACYP2C19
SCHEMBL4948937 0.81 PSMB5 (0.37) POLBPKMPSMB5
SCHEMBL4939631 0.79 MMP2 (0.46) MMP1MMP2MMP9MMP8CNR2
SCHEMBL4949147 0.79 POLB (0.39) POLBPKMGAAMALT1ATM
SCHEMBL4946819 0.77 PSEN1 (0.44)
SCHEMBL4950030 0.75 EP300 (0.37) MMP1MMP2MMP9MMP8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633350-A4 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARM INC (US) 2008-11-26 EP disclosed
EP-1633350-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2006-03-15 EP disclosed
WO-2005009344-A2 ACYLATED AMINO ACID AMIDYL PYRAZOLES AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 2005-02-03 WO disclosed