SCHEMBL4950223

SCHEMBL4950223

CC(=O)Cc1cccc(O[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTBP2 P56545 1/20 0.39
F10 P00742 1/20 0.39
MAOB P27338 1/20 0.38
LTB4R Q15722 1/20 0.38
LTB4R2 Q9NPC1 1/20 0.38
PPARG P37231 2/20 0.36
PPARA Q07869 2/20 0.36
USP2 O75604 1/20 0.36
SLC7A5 Q01650 1/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3978646 0.81 MAOA (0.35) MAOBPPARGPPARAPDK1PDK2
SCHEMBL25456702 0.80 CYSLTR2 (0.50) PPARGPPARACYP1A2
SCHEMBL3321749 0.80 MAOB (0.50) MAOBCYP1A2
SCHEMBL27358205 0.78 AKR1C3 (0.53) PPARGPOLB
SCHEMBL7092637 0.77 CYP3A4 (0.42) POLB
SCHEMBL7805483 0.76 SMN1; SMN2 (0.42) MAOBPOLB
SCHEMBL31139353 0.76 KMT2A (0.56) PPARG
SCHEMBL7221196 0.75 MAOA (0.45) PPARGPPARA
SCHEMBL3319281 0.75 GSK3B (0.49) MAOBPOLB
SCHEMBL10706227 0.75 FFAR1 (0.54) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879886-A1 MITOTIC KINESIN INHIBITORS AND METHODS OF USE THEREOF Array Biopharma, Inc. (US) 2008-01-23 EP disclosed
WO-2006119146-A1 MITOTIC KINESIN INHIBITORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2006-11-09 WO disclosed