SCHEMBL4957415

SCHEMBL4957415

CNC(=O)OCC(Cc1ccc(Cl)c(Cl)c1)c1nnn[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TACR1 P25103 1/20 0.38
PNMT P11086 1/20 0.35
P2RX7 Q99572 1/20 0.34
MAPK1 P28482 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ROCK2 O75116 2/20 0.33
ROCK1 Q13464 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
AURKA O14965 1/20 0.33
DYRK3 O43781 1/20 0.33
PRKD3 O94806 1/20 0.33
PRKCG P05129 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
MARK3 P27448 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4958622 0.89 PSEN1 (0.37) SMN1; SMN2MEN1KMT2AROCK2PSEN1
SCHEMBL4958173 0.85 PNMT (0.38) TSHRSMN1; SMN2TACR1PNMTMAPK1
SCHEMBL17045288 0.76 TSHR (0.51) TSHRSMN1; SMN2TACR1PNMTMAPK1
SCHEMBL17045290 0.76 TSHR (0.51) TSHRSMN1; SMN2TACR1PNMTMAPK1
SCHEMBL17045289 0.76 TSHR (0.51) TSHRSMN1; SMN2TACR1PNMTMAPK1
SCHEMBL4959455 0.73 CYP1A2 (0.42) SMN1; SMN2ROCK2RAB9ANPSR1
SCHEMBL134466 0.71 TSHR (0.57) TSHRSMN1; SMN2TACR1MAPK1MEN1
SCHEMBL4960151 0.70 PNMT (0.40) SMN1; SMN2PNMTKMT2ANPSR1
SCHEMBL10732984 0.70 TSHR (0.55) TSHRSMN1; SMN2TACR1MAPK1MEN1
SCHEMBL4959312 0.70 SLC6A2 (0.43) TSHRSMN1; SMN2TACR1PNMTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1879873-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK Holdings Co., Ltd. (KR) 2008-01-23 EP disclosed
WO-2006112685-A1 NEUROTHERAPEUTIC AZOLE COMPOUNDS SK HOLDINGS CO., LTD. (KR) 2006-10-26 WO disclosed